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TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339102((5-(aminomethyl)-4-(2,4-dichlorophenyl)-6-methylpy...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339100(5-(aminomethyl)-4-(2,4-dichlorophenyl)-6-methylpic...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50229666((2S,3S)-2-((S)-1-((2S,3S)-2-amino-3-methylpentanoy...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339101(5-(aminomethyl)-4-(2,4-dichlorophenyl)-N,6-dimethy...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339103(5-Aminomethyl-4-(2,4-dichlorophenyl)-6-methyl-pyri...)
Affinity DataKi:  6.60E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339095(5-(aminomethyl)-N-cyclopropyl-4-(4-fluorophenyl)-6...)
Affinity DataKi:  1.06E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339096((5-(aminomethyl)-4-(4-fluorophenyl)-6-methylpyridi...)
Affinity DataKi:  1.37E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339099(5-(aminomethyl)-4-(2,4-difluorophenyl)-6-methyl-N-...)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339098(5-(aminomethyl)-N-cyclopropyl-4-(2,4-difluoropheny...)
Affinity DataKi:  1.82E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed