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Found 17 Enz. Inhib. hit(s) with all data for entry = 5798
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94643(1-(3,4-dichlorophenyl)-2-(2-imino-3-prop-2-enyl-1-...)
Affinity DataEC50:  3.33E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM50375133(CHEMBL440586 | cid_703050)
Affinity DataEC50:  2.66E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM64181(4-(7-ethyl-1H-indol-3-yl)-N-(2-methoxyethyl)-1,3-t...)
Affinity DataEC50:  4.88E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94645(MLS-0356781.0001 | N-butan-2-yl-4-(1H-indol-3-yl)-...)
Affinity DataEC50:  7.05E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM51800(4-(1H-indol-3-yl)-N-methyl-1,3-thiazol-2-amine | 4...)
Affinity DataEC50:  1.03E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94646(1-(4-fluorophenyl)-2-(2-imino-3-methyl-1-benzimida...)
Affinity DataEC50:  3.45E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94647(1-(4-chlorophenyl)-2-(2-imino-3-methyl-1-benzimida...)
Affinity DataEC50:  3.09E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94648(1-(3,4-dichlorophenyl)-2-(3-ethyl-2-imino-1-benzim...)
Affinity DataEC50:  2.52E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94649(4-(1H-indol-3-yl)-N-(2-phenylethyl)-1,3-thiazol-2-...)
Affinity DataEC50:  5.13E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94650(4-(7-ethyl-1H-indol-3-yl)-N-prop-2-enyl-1,3-thiazo...)
Affinity DataEC50:  9.24E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM73956(1-(3,4-dichlorophenyl)-2-(2-imino-3-methyl-1-benzi...)
Affinity DataEC50:  2.60E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94651(1-(3,4-dichlorophenyl)-2-[2-imino-3-(phenylmethyl)...)
Affinity DataEC50:  1.55E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94652(1-(3,4-dichlorophenyl)-2-[2-imino-3-(2-pyrrolidin-...)
Affinity DataEC50:  2.42E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94653(4-(1H-indol-3-yl)-N-(1-phenylpropan-2-yl)-1,3-thia...)
Affinity DataEC50:  8.68E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM51920(4-(7-ethyl-1H-indol-3-yl)-N-(1-methoxypropan-2-yl)...)
Affinity DataEC50:  4.56E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94654(4-(1H-indol-3-yl)-N-prop-2-enyl-1,3-thiazol-2-amin...)
Affinity DataEC50:  5.69E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM94644(4-(7-ethyl-1H-indol-3-yl)-N-methyl-1,3-thiazol-2-a...)
Affinity DataEC50:  3.99E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay