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Found 20 Enz. Inhib. hit(s) with all data for entry = 50046105
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094971(CHEMBL3589383)
Affinity DataKi:  12nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094970(CHEMBL3589385)
Affinity DataKi:  14nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094973(CHEMBL3589381)
Affinity DataKi:  18nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50425732(ENZALUTAMIDE | US10053433, FC 4.129 | US10806720, ...)
Affinity DataKi:  28nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094974(CHEMBL3589380)
Affinity DataKi:  34nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094975(956104-40-8 | ARN-509 | JNJ-56021927 | US10053433,...)
Affinity DataKi:  35nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094966(CHEMBL3588961)
Affinity DataKi:  41nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094957(CHEMBL3588965)
Affinity DataKi:  43nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094967(CHEMBL3588960)
Affinity DataKi:  68nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094958(CHEMBL3588959)
Affinity DataKi:  95nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094969(CHEMBL3589387)
Affinity DataKi:  126nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataKi:  160nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094972(CHEMBL3589382)
Affinity DataKi:  215nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094963(CHEMBL3588964)
Affinity DataKi:  236nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094960(CHEMBL3589390)
Affinity DataKi:  257nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094959(CHEMBL3589391)
Affinity DataKi:  482nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094964(CHEMBL3588963)
Affinity DataKi:  515nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094961(CHEMBL3588968)
Affinity DataKi:  576nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094962(CHEMBL3588967)
Affinity DataKi:  585nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094965(CHEMBL3588962)
Affinity DataKi:  798nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed