TargetGlutamate receptor ionotropic, NMDA 2A(Rattus norvegicus (Rat))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataIC50: 3.15E+5nMAssay Description:Agonist activity at rat recombinant NMDA NR2A receptor expressed in xenopus laevis oocyte assessed as inhibition of glycine-stimulated currentMore data for this Ligand-Target Pair
Affinity DataIC50: 3.15E+5nMAssay Description:Agonist activity at rat recombinant NMDA NR1 receptor expressed in xenopus laevis oocyte assessed as inhibition of L-glutamate-stimulated currentMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 3.41E+3nMAssay Description:Agonist activity at mGlu6 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 720nMAssay Description:Agonist activity at mGlu4 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: >3.00E+5nMAssay Description:Agonist activity at mGlu8 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 690nMAssay Description:Agonist activity at mGlu4 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 2.15E+3nMAssay Description:Agonist activity at mGlu8 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 6.51E+3nMAssay Description:Agonist activity at mGlu8 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 1.11E+5nMAssay Description:Agonist activity at mGlu6 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at mGlu4 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 4.08E+4nMAssay Description:Agonist activity at mGlu4 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: >3.00E+6nMAssay Description:Agonist activity at mGlu7 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at mGlu6 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 560nMAssay Description:Agonist activity at mGlu8 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Agonist activity at mGlu8 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 6.25E+5nMAssay Description:Agonist activity at mGlu7 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 6.02E+5nMAssay Description:Agonist activity at mGlu7 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 1.95E+3nMAssay Description:Agonist activity at mGlu6 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at mGlu7 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
University Paris Descartes
Curated by ChEMBL
University Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 1.85E+3nMAssay Description:Agonist activity at mGlu4 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate productionMore data for this Ligand-Target Pair