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Found 76 Enz. Inhib. hit(s) with all data for entry = 50027742
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266136((R)-3-(4-iodobenzylthio)-2-((S)-3-mercapto-2-methy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266170((R)-3-(4-ethylbenzylthio)-2-((S)-3-mercapto-2-meth...)
Affinity DataIC50:  21nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266173((R)-3-(4-tert-butylbenzylthio)-2-((S)-3-mercapto-2...)
Affinity DataIC50:  24nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266075((R)-3-(benzylthio)-2-((S)-3-mercapto-2-methylpropa...)
Affinity DataIC50:  34nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266244((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(m...)
Affinity DataIC50:  46nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266316((R)-3-(2-(4-cyclohexylphenyl)propan-2-ylthio)-2-((...)
Affinity DataIC50:  55nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266247((2R)-3-(1-(4-isopropylphenyl)ethylthio)-2-((S)-3-m...)
Affinity DataIC50:  55nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266248((2R)-3-(1-(4-isopropylphenyl)propylthio)-2-((S)-3-...)
Affinity DataIC50:  67nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266171((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-pr...)
Affinity DataIC50:  72nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266175((R)-3-(4-cyclohexylbenzylthio)-2-((S)-3-mercapto-2...)
Affinity DataIC50:  79nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266280((R)-3-(2-(4-isopropylphenyl)propan-2-ylthio)-2-((S...)
Affinity DataIC50:  79nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266279((2R)-3-((4-isopropylphenyl)(phenyl)methylthio)-2-(...)
Affinity DataIC50:  91nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266208((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-me...)
Affinity DataIC50:  100nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266133((R)-3-(4-fluorobenzylthio)-2-((S)-3-mercapto-2-met...)
Affinity DataIC50:  100nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266173((R)-3-(4-tert-butylbenzylthio)-2-((S)-3-mercapto-2...)
Affinity DataIC50:  130nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266136((R)-3-(4-iodobenzylthio)-2-((S)-3-mercapto-2-methy...)
Affinity DataIC50:  140nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266138((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(t...)
Affinity DataIC50:  140nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266245((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(m...)
Affinity DataIC50:  158nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266276((2R)-3-(1-(4-isopropylphenyl)butylthio)-2-((S)-3-m...)
Affinity DataIC50:  180nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266172((R)-3-(4-isopropylbenzylthio)-2-((S)-3-mercapto-2-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266247((2R)-3-(1-(4-isopropylphenyl)ethylthio)-2-((S)-3-m...)
Affinity DataIC50:  200nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266315((2R)-3-((4-cyclohexylphenyl)(phenyl)methylthio)-2-...)
Affinity DataIC50:  210nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266171((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-pr...)
Affinity DataIC50:  210nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266137((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-me...)
Affinity DataIC50:  240nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266134((R)-3-(4-chlorobenzylthio)-2-((S)-3-mercapto-2-met...)
Affinity DataIC50:  250nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266209((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(t...)
Affinity DataIC50:  260nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266280((R)-3-(2-(4-isopropylphenyl)propan-2-ylthio)-2-((S...)
Affinity DataIC50:  260nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266174((R)-3-(biphenyl-4-ylmethylthio)-2-((S)-3-mercapto-...)
Affinity DataIC50:  280nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266170((R)-3-(4-ethylbenzylthio)-2-((S)-3-mercapto-2-meth...)
Affinity DataIC50:  280nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266135((R)-3-(4-bromobenzylthio)-2-((S)-3-mercapto-2-meth...)
Affinity DataIC50:  280nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266213((R)-3-(4-cyanobenzylthio)-2-((S)-3-mercapto-2-meth...)
Affinity DataIC50:  300nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266245((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(m...)
Affinity DataIC50:  300nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266244((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(m...)
Affinity DataIC50:  300nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266172((R)-3-(4-isopropylbenzylthio)-2-((S)-3-mercapto-2-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266243((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-ni...)
Affinity DataIC50:  320nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266210((R)-3-(4-ethoxybenzylthio)-2-((S)-3-mercapto-2-met...)
Affinity DataIC50:  340nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266248((2R)-3-(1-(4-isopropylphenyl)propylthio)-2-((S)-3-...)
Affinity DataIC50:  340nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266138((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(t...)
Affinity DataIC50:  340nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266211((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-ph...)
Affinity DataIC50:  370nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266209((R)-2-((S)-3-mercapto-2-methylpropanamido)-3-(4-(t...)
Affinity DataIC50:  400nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266276((2R)-3-(1-(4-isopropylphenyl)butylthio)-2-((S)-3-m...)
Affinity DataIC50:  420nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266277((2R)-3-(1-(4-isopropylphenyl)-2-methylpropylthio)-...)
Affinity DataIC50:  430nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266079((R)-3-(4-(dimethylamino)benzylthio)-2-(2-mercaptoa...)
Affinity DataIC50:  470nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266278((2R)-3-(1-(4-isopropylphenyl)pentylthio)-2-((S)-3-...)
Affinity DataIC50:  510nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266074(CHEMBL457317 | S-(4-dimethylamino)benzy-N-[(2S)-3-...)
Affinity DataIC50:  520nMAssay Description:Inhibition of angiotensin-converting enzyme (unknown origin) in whole blood by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266277((2R)-3-(1-(4-isopropylphenyl)-2-methylpropylthio)-...)
Affinity DataIC50:  520nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266213((R)-3-(4-cyanobenzylthio)-2-((S)-3-mercapto-2-meth...)
Affinity DataIC50:  525nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266174((R)-3-(biphenyl-4-ylmethylthio)-2-((S)-3-mercapto-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266135((R)-3-(4-bromobenzylthio)-2-((S)-3-mercapto-2-meth...)
Affinity DataIC50:  610nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene A-4 hydrolase(Cavia porcellus)
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50266210((R)-3-(4-ethoxybenzylthio)-2-((S)-3-mercapto-2-met...)
Affinity DataIC50:  640nMAssay Description:Inhibition of LTA4 hydrolase in guinea pig lung assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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