Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50030492
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296994(CHEMBL561939 | N-(5-Methanesulfonylamino-4,6-dimet...)
Affinity DataIC50:  13nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50263150(CHEMBL513892 | N-(4,6-dimethyl-1-octylindolin-7-yl...)
Affinity DataIC50:  24nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297009(CHEMBL550526 | N-(1-decyl-4,6-dimethylindolin-7-yl...)
Affinity DataIC50:  27nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297008(CHEMBL558454 | N-(1-heptyl-4,6-dimethylindolin-7-y...)
Affinity DataIC50:  30nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297017(CHEMBL555564 | N-[1-(Cyclobutylmethyl)-5-methanesu...)
Affinity DataIC50:  36nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297014(CHEMBL559117 | N-[5-Methanesulfonylamino-4,6-dimet...)
Affinity DataIC50:  40nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296993(CHEMBL557522 | N-(1-Hexyl-5-methanesulfonylamino-4...)
Affinity DataIC50:  42nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296992(CHEMBL559879 | N-(5-Methanesulfonylamino-4,6-dimet...)
Affinity DataIC50:  49nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297022(CHEMBL564138 | N-(1-Butyl-5-methanesulfonylamino-4...)
Affinity DataIC50:  53nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297010(CHEMBL561477 | N-(1-dodecyl-4,6-dimethylindolin-7-...)
Affinity DataIC50:  58nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297013(CHEMBL554505 | N-[1-(2,2-Dimethylpropyl)-5-methane...)
Affinity DataIC50:  61nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297007(CHEMBL561074 | N-(1-hexyl-4,6-dimethylindolin-7-yl...)
Affinity DataIC50:  67nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297015(CHEMBL559318 | N-[5-Methanesulfonylamino-4,6-dimet...)
Affinity DataIC50:  68nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296991(CHEMBL551271 | N-(1-Butyl-5-methanesulfonylamino-4...)
Affinity DataIC50:  69nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297012(CHEMBL549649 | N-[5-Methanesulfonylamino-4,6-dimet...)
Affinity DataIC50:  71nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297018(CHEMBL556503 | N-[1-(Cyclopentyl)-5-methanesulfony...)
Affinity DataIC50:  95nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297006(CHEMBL563443 | N-(4,6-dimethyl-1-pentylindolin-7-y...)
Affinity DataIC50:  110nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297025(CHEMBL561135 | N-(5,7-dimethyl-6-(methylsulfonamid...)
Affinity DataIC50:  130nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297016(CHEMBL560997 | N-[1-(Cyclopropylmethyl)-5-methanes...)
Affinity DataIC50:  160nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297005(CHEMBL538381 | N-(1-butyl-4,6-dimethylindolin-7-yl...)
Affinity DataIC50:  220nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296990(CHEMBL559348 | N-(5-Methanesulfonylamino-4,6-dimet...)
Affinity DataIC50:  240nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297023(CHEMBL556232 | N-(1-Butyl-5-methanesulfonylamino-4...)
Affinity DataIC50:  240nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297019(CHEMBL551410 | N-[5-Methanesulfonylamino-1-(2-meth...)
Affinity DataIC50:  270nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297020(CHEMBL563918 | N-[1-(2-Ethoxyethyl)-5-methanesulfo...)
Affinity DataIC50:  310nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297024(CHEMBL563699 | N-(1-Isobutyl-5-methanesulfonylamin...)
Affinity DataIC50:  480nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297004(CHEMBL554163 | N-(4,6-dimethyl-1-propylindolin-7-y...)
Affinity DataIC50:  570nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296999(CHEMBL549714 | [1-Decyl-7-(2,2-dimethylpropanamido...)
Affinity DataIC50:  910nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297000(CHEMBL563263 | [7-(2,2-Dimethylpropanamido)-4,6-di...)
Affinity DataIC50:  960nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297001(CHEMBL564069 | [7-(2,2-Dimethylpropanamido)-1-dode...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296998(CHEMBL558325 | [7-(2,2-Dimethylpropanamido)-4,6-di...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296989(CHEMBL561798 | N-(1-Ethyl-5-methanesulfonylamino-4...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50263192(CHEMBL478858 | CHEMBL564483 | Pactimibe | [7-(2,2-...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297021(CHEMBL558831 | N-(1-Butyl-5-methanesulfonylamino-4...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297011(CHEMBL558455 | N-(1-Isopropyl-5-methanesulfonylami...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297003(CHEMBL558062 | N-(1-ethyl-4,6-dimethylindolin-7-yl...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296995(CHEMBL557933 | [7-(2,2-Dimethylpropanamido)-1-hexy...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296996(CHEMBL551676 | [7-(2,2-Dimethylpropanamido)-1-hept...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50296988(CHEMBL562996 | N-(5-Methanesulfonylamino-1,4,6-tri...)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50297002(CHEMBL564833 | N-(1,4,6-trimethylindolin-7-yl)piva...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed