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Found 7 Enz. Inhib. hit(s) with all data for entry = 50048329
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.300nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50212821(CHEMBL3301661)
Affinity DataKi:  4.60nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
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TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50212820(BMY-20014 | CHEMBL151910)
Affinity DataKi:  13nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
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TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50212823(BMY-42803 | BMY-42804 | CHEMBL2115538)
Affinity DataKi:  36nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
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TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50212822(CHEMBL2111202)
Affinity DataKi: >1.00E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50212824(CHEMBL2111260)
Affinity DataKi: >1.00E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50101817(Adalat | Adalat Cc | Afeditab Cr | BAY-A-1040 | CH...)
Affinity DataKi: >1.00E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails