Compile Data Set for Download or QSAR
maximum 50k data
Found 35 Enz. Inhib. hit(s) with all data for entry = 50035476
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367049(CHEMBL604399)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367049(CHEMBL604399)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367044(CHEMBL605639)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of AMP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367044(CHEMBL605639)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367040(CHEMBL606017)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367040(CHEMBL606017)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367048(CHEMBL605430)
Affinity DataKi:  5.20E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367048(CHEMBL605430)
Affinity DataKi:  6.30E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP,competitive and non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010309(CHEMBL3251358)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM18137(AMP | CHEMBL752 | US11185100, TABLE 7.3 | [(2R,3S,...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366480(ADENOSINE TRIPHOSPHATE | ATP)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367038(CHEMBL604815)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of AMP competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367038(CHEMBL604815)
Affinity DataKi:  4.50E+5nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP,competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367046(CHEMBL604395)
Affinity DataKi:  4.50E+5nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367042(CHEMBL606221)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366480(ADENOSINE TRIPHOSPHATE | ATP)
Affinity DataKi:  5.70E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM18137(AMP | CHEMBL752 | US11185100, TABLE 7.3 | [(2R,3S,...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of AMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367039(CHEMBL604398)
Affinity DataKi:  1.80E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367037(CHEMBL606008)
Affinity DataKi:  1.80E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367037(CHEMBL606008)
Affinity DataKi:  2.00E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP,competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367039(CHEMBL604398)
Affinity DataKi:  2.20E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367045(CHEMBL605010)
Affinity DataKi:  3.20E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367042(CHEMBL606221)
Affinity DataKi:  4.00E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATP non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367046(CHEMBL604395)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATPnon competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367045(CHEMBL605010)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010309(CHEMBL3251358)
Affinity DataKi:  6.10E+6nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme in the presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367041(CHEMBL603556)
Affinity DataKi:  9.80E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367047(CHEMBL2368667)
Affinity DataKi:  1.50E+7nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367041(CHEMBL603556)
Affinity DataKi:  1.60E+7nMAssay Description:Inhibitory activity against rat Adenylate kinase M isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  1.90E+7nMAssay Description:Inhibitory activity against rat adenylate kinase II (AK-II) isoenzyme was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367047(CHEMBL2368667)
Affinity DataKi:  2.10E+7nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase isoenzyme 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  8.20E+7nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  8.70E+7nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  9.20E+7nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed