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Found 122 Enz. Inhib. hit(s) with all data for entry = 50018195
LigandPNGBDBM466723(US10800761, Example 42 | US10800761, Example 55 | ...)
Affinity DataKi: <0.100nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50405899(CHEMBL5288420)
Affinity DataKi: <1nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
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LigandPNGBDBM466728(US10800761, Example 47 | US11731958, Example 47)
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM466724(US10800761, Example 43 | US11731958, Example 43)
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM466705(US10800761, Example 24)
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50406012(CHEMBL5273201)
Affinity DataKi:  1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM50406009(CHEMBL5284132)
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM50405947(CHEMBL5274764)
Affinity DataKi:  1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM459445(US10752635, Example 5, Peak 1 | US11492354, Exampl...)
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50406013(CHEMBL5267188)
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM50405898(CHEMBL5283973)
Affinity DataKi: <1nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
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LigandPNGBDBM50405897(CHEMBL5277241)
Affinity DataKi: <1nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
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LigandPNGBDBM50405896(CHEMBL5281003)
Affinity DataKi: <1nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
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LigandPNGBDBM459444(US10752635, Example 4, Peak 2 | US11492354, Exampl...)
Affinity DataKi: <1nMAssay Description:Antihistaminic activity against Histamine H1 receptor was measured on isolated terminal part of guinea pig ileumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM459443(US10752635, Example 4, Peak 1 | US11492354, Exampl...)
Affinity DataKi:  1nMAssay Description:Antihistaminic activity against Histamine H1 receptor was measured on isolated terminal part of guinea pig ileumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50405892(CHEMBL5267747)
Affinity DataKi: <1nMAssay Description:Antihistaminic activity against Histamine H1 receptor was measured on isolated terminal part of guinea pig ileumMore data for this Ligand-Target Pair
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LigandPNGBDBM50406008(CHEMBL5276026)
Affinity DataKi:  1.5nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM50405900(CHEMBL5268277)
Affinity DataKi:  1.60nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
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LigandPNGBDBM466704(US10800761, Example 23 | US11731958, Example 23)
Affinity DataKi:  1.70nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM459439(US10752635, Example 1, Peak 2 | US11492354, Exampl...)
Affinity DataKi:  1.80nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM466687(US10800761, Example 6 | US11731958, Example 6 | US...)
Affinity DataKi:  1.90nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50405895(CHEMBL5279971)
Affinity DataKi:  2nMAssay Description:Vasopressin V2 receptor antagonistic activity in vivo in anesthetized ratsMore data for this Ligand-Target Pair
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LigandPNGBDBM466727(US10800761, Example 46 | US11731958, Example 46)
Affinity DataKi:  2nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM466682(US10800761, Example 1 | US11731958, Example 1)
Affinity DataKi:  2.20nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM459441(US10752635, Example 3, Peak 1 | US11492354, Exampl...)
Affinity DataKi:  2.20nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM459484(US10752635, Example 35 | US11492354, Example 35)
Affinity DataKi:  2.20nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50405893(CHEMBL5271378)
Affinity DataKi:  2.60nMAssay Description:Antihistaminic activity against Histamine H1 receptor was measured on isolated terminal part of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50405894(CHEMBL5269770)
Affinity DataKi:  3nMAssay Description:Antihistaminic activity against Histamine H1 receptor was measured on isolated terminal part of guinea pig ileumMore data for this Ligand-Target Pair
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LigandPNGBDBM50405946(CHEMBL5279231)
Affinity DataKi:  3.30nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM50406004(CHEMBL5267479)
Affinity DataKi:  3.90nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM50406010(CHEMBL5277513)
Affinity DataKi:  7.10nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM50405891(CHEMBL5290431)
Affinity DataKi:  22nMAssay Description:Antihistaminic activity against Histamine H1 receptor was measured on isolated terminal part of guinea pig ileumMore data for this Ligand-Target Pair
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LigandPNGBDBM50405897(CHEMBL5277241)
Affinity DataKi:  23nMAssay Description:Antagonistic activity against Thromboxane A2 receptor in guinea pig trachea in the presence of 11,9-epoxymethano-PGH2More data for this Ligand-Target Pair
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LigandPNGBDBM50405896(CHEMBL5281003)
Affinity DataKi:  36nMAssay Description:Antagonistic activity against Thromboxane A2 receptor in guinea pig trachea in the presence of 9,11-azo-PGH2More data for this Ligand-Target Pair
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LigandPNGBDBM466723(US10800761, Example 42 | US10800761, Example 55 | ...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50405895(CHEMBL5279971)
Affinity DataKi:  64nMAssay Description:Antagonistic activity against Thromboxane A2 receptor in rat aorta in the presence of 11,9-epoxymethano-PGH2More data for this Ligand-Target Pair
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LigandPNGBDBM50406013(CHEMBL5267188)
Affinity DataKi:  65nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
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LigandPNGBDBM466728(US10800761, Example 47 | US11731958, Example 47)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM459444(US10752635, Example 4, Peak 2 | US11492354, Exampl...)
Affinity DataKi:  100nMAssay Description:Antagonistic activity against Thromboxane A2 receptor in rat aorta in the presence of 11,9-epoxymethano-PGH2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM459443(US10752635, Example 4, Peak 1 | US11492354, Exampl...)
Affinity DataKi:  105nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM466724(US10800761, Example 43 | US11731958, Example 43)
Affinity DataKi:  124nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM466705(US10800761, Example 24)
Affinity DataKi:  129nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50405894(CHEMBL5269770)
Affinity DataKi:  211nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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LigandPNGBDBM466727(US10800761, Example 46 | US11731958, Example 46)
Affinity DataKi:  232nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50406012(CHEMBL5273201)
Affinity DataKi:  270nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
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LigandPNGBDBM466704(US10800761, Example 23 | US11731958, Example 23)
Affinity DataKi:  276nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM466687(US10800761, Example 6 | US11731958, Example 6 | US...)
Affinity DataKi:  356nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50406010(CHEMBL5277513)
Affinity DataKi:  408nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
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LigandPNGBDBM466682(US10800761, Example 1 | US11731958, Example 1)
Affinity DataKi:  541nMAssay Description:Inhibitory activity against human carbonic anhydrase II using pH stat assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50405893(CHEMBL5271378)
Affinity DataKi:  1.11E+3nMAssay Description:In vitro inhibition of human carbonic anhydrase II (0.1 nM).More data for this Ligand-Target Pair
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