Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50001669
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291987(CHEMBL4160562)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291965(CHEMBL4163356)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291986(CHEMBL4167795)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291964(CHEMBL4174712)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291963(CHEMBL4166811)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291982(CHEMBL4175661)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291992(CHEMBL4160951)
Affinity DataIC50:  18nMAssay Description:Inhibition of VCAM (vascular cell adhesion molecule) adhesion to alpha4-beta1 integrin of leukocyte cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291988(CHEMBL4171159)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291967(CHEMBL4159993)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291975(CHEMBL4167914)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292173(CHEMBL4162019)
Affinity DataIC50:  21nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291966(CHEMBL4171262)
Affinity DataIC50:  26nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292156(CHEMBL4172245)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292172(CHEMBL4164355)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50291991(CHEMBL4168889)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292234(CHEMBL4164636)
Affinity DataIC50:  37nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292218(CHEMBL4169134)
Affinity DataIC50:  46nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292232(CHEMBL4176144)
Affinity DataIC50:  46nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292233(CHEMBL4175919)
Affinity DataIC50:  52nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292206(CHEMBL4161215)
Affinity DataIC50:  58nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292181(CHEMBL4172683)
Affinity DataIC50:  67nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50292231(CHEMBL4172516)
Affinity DataIC50:  116nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  176nMAssay Description:Inhibition of recombinant wild type HIV1 reverse transcriptase p66/p51 using poly (rA)/anoligo (dT)16 as template/primer assessed as inhibition of bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed