Affinity DataIC50: 37nMAssay Description:Antagonist activity at P2Y6 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Antagonist activity at P2Y1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 148nMAssay Description:Antagonist activity at P2Y1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Antagonist activity at P2Y1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Agonist activity at P2Y2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.25E+3nMAssay Description:Agonist activity at P2Y2 receptor in NG108-15 cells (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at P2Y2 receptor in human CF/T43 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Agonist activity at P2Y2 receptor in BEA cells (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.72E+3nMAssay Description:Agonist activity at human N-terminal HA-tagged P2Y2 receptor expressed in 1321N1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 3.78E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 2.63E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 47nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 103nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Agonist activity at P2Y2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 4.89E+5nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Agonist activity at P2Y2 receptor in NG108-15 cells (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 710nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at P2Y2 receptor (unknown origin) expressed in human 1321N1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 840nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at P2Y2 receptor in human CF/T43 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at P2Y2 receptor in BEA cells (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.98E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 187nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Agonist activity at P2Y2 receptor (unknown origin) assessed as reduction in inositol phosphate accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 109nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 139nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 1.55E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as [3H]-inositol phosphate accumulation measured after 90 mins by anion ex...More data for this Ligand-Target Pair