Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 3224
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29563(1-(m-trifluorophenyl)piperazine, 10)
Affinity DataKi:  0.300nM ΔG°:  -56.5kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29567(1-(m-trifluorophenyl)piperazine, 14)
Affinity DataKi:  1.30nM ΔG°:  -52.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29565(1-(m-trifluorophenyl)piperazine, 12)
Affinity DataKi:  1.5nM ΔG°:  -52.4kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29566(1-(m-trifluorophenyl)piperazine, 13)
Affinity DataKi:  2.20nM ΔG°:  -51.4kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29561(1-(m-trifluorophenyl)piperazine, 8)
Affinity DataKi:  2.60nM ΔG°:  -51.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29560(1-(m-trifluorophenyl)piperazine, 7)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29558(1-(m-trifluorophenyl)piperazine, 5)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29557(1-(m-trifluorophenyl)piperazine, 4)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29563(1-(m-trifluorophenyl)piperazine, 10)
Affinity DataKi:  4nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29562(1-(m-trifluorophenyl)piperazine, 9)
Affinity DataKi:  5.90nM ΔG°:  -48.9kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29559(1-(m-trifluorophenyl)piperazine, 6)
Affinity DataKi:  9nM ΔG°:  -47.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29560(1-(m-trifluorophenyl)piperazine, 7)
Affinity DataKi:  21nM ΔG°:  -45.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29556(1-(m-trifluorophenyl)piperazine, 3)
Affinity DataKi:  21nM ΔG°:  -45.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29567(1-(m-trifluorophenyl)piperazine, 14)
Affinity DataKi:  24nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29562(1-(m-trifluorophenyl)piperazine, 9)
Affinity DataKi:  30nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29564(1-(m-trifluorophenyl)piperazine, 11)
Affinity DataKi:  31nM ΔG°:  -44.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29564(1-(m-trifluorophenyl)piperazine, 11)
Affinity DataKi:  34nM ΔG°:  -44.3kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29565(1-(m-trifluorophenyl)piperazine, 12)
Affinity DataKi:  43nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29558(1-(m-trifluorophenyl)piperazine, 5)
Affinity DataKi:  46nM ΔG°:  -43.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29566(1-(m-trifluorophenyl)piperazine, 13)
Affinity DataKi:  48nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29564(1-(m-trifluorophenyl)piperazine, 11)
Affinity DataKi:  73nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29561(1-(m-trifluorophenyl)piperazine, 8)
Affinity DataKi:  85nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29560(1-(m-trifluorophenyl)piperazine, 7)
Affinity DataKi:  101nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29566(1-(m-trifluorophenyl)piperazine, 13)
Affinity DataKi:  107nM ΔG°:  -41.4kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29558(1-(m-trifluorophenyl)piperazine, 5)
Affinity DataKi:  127nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29556(1-(m-trifluorophenyl)piperazine, 3)
Affinity DataKi:  128nM ΔG°:  -40.9kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29562(1-(m-trifluorophenyl)piperazine, 9)
Affinity DataKi:  134nM ΔG°:  -40.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29559(1-(m-trifluorophenyl)piperazine, 6)
Affinity DataKi:  221nM ΔG°:  -39.5kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29559(1-(m-trifluorophenyl)piperazine, 6)
Affinity DataKi:  268nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29565(1-(m-trifluorophenyl)piperazine, 12)
Affinity DataKi:  335nM ΔG°:  -38.4kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29556(1-(m-trifluorophenyl)piperazine, 3)
Affinity DataKi:  483nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29557(1-(m-trifluorophenyl)piperazine, 4)
Affinity DataKi:  505nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29561(1-(m-trifluorophenyl)piperazine, 8)
Affinity DataKi:  1.20E+3nM ΔG°:  -35.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29557(1-(m-trifluorophenyl)piperazine, 4)
Affinity DataKi:  1.82E+3nM ΔG°:  -34.1kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29558(1-(m-trifluorophenyl)piperazine, 5)
Affinity DataKi:  2.34E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29563(1-(m-trifluorophenyl)piperazine, 10)
Affinity DataKi:  2.64E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29564(1-(m-trifluorophenyl)piperazine, 11)
Affinity DataKi:  2.72E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29567(1-(m-trifluorophenyl)piperazine, 14)
Affinity DataKi:  3.60E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29566(1-(m-trifluorophenyl)piperazine, 13)
Affinity DataKi:  4.37E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29565(1-(m-trifluorophenyl)piperazine, 12)
Affinity DataKi:  4.68E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29560(1-(m-trifluorophenyl)piperazine, 7)
Affinity DataKi: >5.00E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29561(1-(m-trifluorophenyl)piperazine, 8)
Affinity DataKi: >5.00E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29562(1-(m-trifluorophenyl)piperazine, 9)
Affinity DataKi: >5.00E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29567(1-(m-trifluorophenyl)piperazine, 14)
Affinity DataKi: >5.00E+3nM ΔG°: >-31.5kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Polish Academy of Sciences

LigandPNGBDBM29563(1-(m-trifluorophenyl)piperazine, 10)
Affinity DataKi: >5.00E+3nM ΔG°: >-31.5kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29559(1-(m-trifluorophenyl)piperazine, 6)
Affinity DataKi: >1.00E+4nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29557(1-(m-trifluorophenyl)piperazine, 4)
Affinity DataKi: >2.50E+4nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Polish Academy of Sciences

LigandPNGBDBM29556(1-(m-trifluorophenyl)piperazine, 3)
Affinity DataKi: >3.00E+4nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed