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Found 16 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 3521
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35890(flufenamic acid analogue, 17)
Affinity DataIC50:  4.40E+3nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35885(flufenamic acid tricyclic analogue, 9)
Affinity DataIC50:  1.03E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50:  1.20E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35897(flufenamic acid analogue, 24)
Affinity DataIC50:  1.35E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35909(2-Hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-ph...)
Affinity DataIC50:  3.30E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35900(flufenamic acid analogue, 27)
Affinity DataIC50:  3.70E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35901(cid_201986 | flufenamic acid analogue, 28)
Affinity DataIC50:  3.70E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35905(Tolfenamic acid | cid_610479 | flufenamic acid ana...)
Affinity DataIC50:  5.79E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35886(flufenamic acid tricyclic analogue, 11)
Affinity DataIC50:  6.75E+4nMpH: 7.2 T: 2°CAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35914(flufenamic acid analogue, 40)
Affinity DataEC50:  5.40E+4nMAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35908(flufenamic acid analogue, 35 | flufenamic acid ana...)
Affinity DataEC50:  5.60E+4nMAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35916(flufenamic acid analogue, 42)
Affinity DataEC50:  6.40E+4nMAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35917(flufenamic acid analogue, 43)
Affinity DataEC50:  7.55E+4nMAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35918(flufenamic acid analogue, 44)
Affinity DataEC50:  8.30E+4nMAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35919(flufenamic acid analogue, 45)
Affinity DataEC50:  9.30E+4nMAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataEC50:  6.70E+4nMAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair