Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50008209
TargetAndrogen receptor(Rattus norvegicus (Rat))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50516763(CHEMBL3185021)
Affinity DataIC50:  36nMAssay Description:Antagonist activity at GAL4-DBD fused rat androgen receptor expressed in UAS-bla 293 cells assessed as reduction in R1881-induced activation incubate...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50:  490nMAssay Description:Antagonist activity at GAL4-DBD fused rat androgen receptor expressed in UAS-bla 293 cells assessed as reduction in R1881-induced activation incubate...More data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50516764(CHEMBL4473164)
Affinity DataIC50:  540nMAssay Description:Antagonist activity at GAL4-DBD fused rat androgen receptor expressed in UAS-bla 293 cells assessed as reduction in R1881-induced activation incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50516765(CHEMBL4581912)
Affinity DataIC50:  1.81E+3nMAssay Description:Antagonist activity at GAL4-DBD fused rat androgen receptor expressed in UAS-bla 293 cells assessed as reduction in R1881-induced activation incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed