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Found 20 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50040377
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393265(CHEMBL2152016)
Affinity DataKi:  540nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393263(CHEMBL2152014)
Affinity DataKi:  540nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273444(CHEMBL463976 | N-Phenyl-2-(pyridin-4-yl)quinoline-...)
Affinity DataKi:  700nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393264(CHEMBL2152015)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393273(CHEMBL2152024)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393275(CHEMBL2152026)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393272(CHEMBL2152023)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393276(CHEMBL2151049)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393259(CHEMBL2152010)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393268(CHEMBL2152019)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393262(CHEMBL2152013)
Affinity DataKi:  3.97E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393261(CHEMBL2152012)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393271(CHEMBL2152022)
Affinity DataKi:  6.90E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393274(CHEMBL2152025)
Affinity DataKi:  8.40E+3nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393266(CHEMBL2152017)
Affinity DataKi:  1.19E+4nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393260(CHEMBL2152011)
Affinity DataKi:  1.44E+4nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273446(CHEMBL513115 | N-Phenyl-2-(pyridin-2-yl)quinoline-...)
Affinity DataKi:  1.45E+4nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393270(CHEMBL2152021)
Affinity DataKi:  1.59E+4nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393269(CHEMBL2152020)
Affinity DataKi:  2.01E+4nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50393267(CHEMBL2152018)
Affinity DataKi:  3.29E+4nMAssay Description:Inhibition of recombinant CYP3A4 NF-14 expressed in Escherichia coli assessed as formation of 6-beta-hydroxytestosterone using testosterone as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed