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Found 10 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 9287
TargetGalectin-3(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455401(3,3'-Dideoxy-3- [4-(morpholin-4- yl)-1H-1,2,3- tri...)
Affinity DataKd:  2nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455401(3,3'-Dideoxy-3- [4-(morpholin-4- yl)-1H-1,2,3- tri...)
Affinity DataKd:  110nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455402(3,3′-Dideoxy-3-[4-(4-methylpiperazin-1-yl)-1...)
Affinity DataKd:  7nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455402(3,3′-Dideoxy-3-[4-(4-methylpiperazin-1-yl)-1...)
Affinity DataKd:  35nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455405(3,3′-Dideoxy-3-[4-(propan-2-yl)-1H-1,2,3-tri...)
Affinity DataKd:  70nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455403(3,3′-Dideoxy-3-[4-(piperidin-4-yl)-1H-1,2,3-...)
Affinity DataKd:  29nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455404(3,3′-Dideoxy-3-[4-(tetrahydropyran-4-yl)-1H-...)
Affinity DataKd:  1nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-1(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455404(3,3′-Dideoxy-3-[4-(tetrahydropyran-4-yl)-1H-...)
Affinity DataKd:  58nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455405(3,3′-Dideoxy-3-[4-(propan-2-yl)-1H-1,2,3-tri...)
Affinity DataKd:  2nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Galecto Biotech

US Patent
LigandPNGBDBM455403(3,3′-Dideoxy-3-[4-(piperidin-4-yl)-1H-1,2,3-...)
Affinity DataKd:  5nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent