Affinity DataIC50: 1.5nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as suppression of [35S]GTPgammaS binding incubated for 60 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as suppression of [35S]GTPgammaS binding incubated for 60 ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as suppression of [35S]GTPgammaS binding incubated for 60 ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as suppression of [35S]GTPgammaS binding incubated for 60 ...More data for this Ligand-Target Pair