BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50047332

Proteasome subunit beta type-5(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

BDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)

IC50: 1.90nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome using ZGlyGlyLeuAMC/SucLeuLeuValTyrAMC as substrate measured every minute for 25 min...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article PubMed DrugBank
PDB

3D Structure (crystal)