BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with all data for assayid = 20 entry = 50002119

Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL

BDBM50370385((R)-TIPIFARNIB | R-11577 | R-115777 | Tipifarnib |...)

IC50: 7.90nMAssay Description:Inhibition of FTase isolated from Kirsten virus-transformed human osteosarcoma cells using K-rasB peptide as substrate in presence of [3H]farnesyl PP...More data for this Ligand-Target Pair

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3D Structure (crystal)