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Found 8 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50033190
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50:  1.20E+4nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341143((E)-2-(3-(3-(2-(4-methylbenzoyl)-1H-imidazol-1-yl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341144((E)-2-(3-(3-(2-(4-methylbenzoyl)-1H-benzo[d]imidaz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341149((E)-2-methyl-2-(3-(2-(2-(4-methylbenzoyl)-1H-benzo...)
Affinity DataEC50:  2.40E+3nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341146((E)-2-(3-(3-(4,5-dimethyl-2-(4-methylbenzoyl)-1H-i...)
Affinity DataEC50:  3.60E+3nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341147((E)-2-methyl-2-(3-(3-(2-(4-methylbenzoyl)-4,5,6,7-...)
Affinity DataEC50:  3.60E+3nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341148((E)-2-methyl-2-(3-(3-(2-(4-methylbenzoyl)-1H-benzo...)
Affinity DataEC50:  3.60E+3nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341145((E)-2-methyl-2-(3-(3-(2-(4-methylbenzoyl)-1H-imida...)
Affinity DataEC50:  620nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells cotransfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed