Affinity DataEC50: 590nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cells co-expressing Galphaq16 assessed as inhibition of calcium mobilization after...More data for this Ligand-Target Pair
Affinity DataEC50: 586nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cells co-expressing Galphaq16 assessed as inhibition of calcium mobilization after...More data for this Ligand-Target Pair