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Found 2 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50002817
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50463401(CHEMBL4242565)
Affinity DataEC50:  590nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cells co-expressing Galphaq16 assessed as inhibition of calcium mobilization after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataEC50:  586nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in HEK293 cells co-expressing Galphaq16 assessed as inhibition of calcium mobilization after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank