Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50043707
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology

Curated by ChEMBL
LigandPNGBDBM50444909(CHEMBL3099618)
Affinity DataKi:  340nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology

Curated by ChEMBL
LigandPNGBDBM50444908(CHEMBL3099624)
Affinity DataKi:  670nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology

Curated by ChEMBL
LigandPNGBDBM50444888(CHEMBL3099621)
Affinity DataKi:  1.02E+3nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed