Compile Data Set for Download or QSAR
Report error Found 234 of kd data for polymerid = 2129,5536,5768,49000132,49000137,49000138,50001754
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207816BDBM50207816(N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3...)
Affinity DataKd:  0.170nMAssay Description:Binding affinity to human adenosine A1 receptor assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095602BDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.240nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor(AR) at 0.1 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095602BDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.260nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.05 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095604BDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.270nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.1 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095604BDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.280nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 0.05 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095602BDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.310nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 100 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095606BDBM50095606(4-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahy...)
Affinity DataKd:  0.320nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039676BDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.330nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039676BDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.330nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039676BDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.330nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095604BDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.340nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095602BDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor(AR) at 5 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095602BDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095602BDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095604BDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.370nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095605BDBM50095605(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.370nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120223BDBM50120223(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.400nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120223BDBM50120223(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.400nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024563BDBM50024563(CHEMBL3330574)
Affinity DataKd:  0.460nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120221BDBM50120221(4-[5-(8-Bicyclo[2.2.1]hept-2-yl-2,6-dioxo-1-propyl...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120221BDBM50120221(4-[5-(8-Bicyclo[2.2.1]hept-2-yl-2,6-dioxo-1-propyl...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120222BDBM50120222(4-[5-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120222BDBM50120222(4-[5-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039675BDBM50039675(3-[(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-p...)
Affinity DataKd:  0.690nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039675BDBM50039675(3-[(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-p...)
Affinity DataKd:  0.690nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039674BDBM50039674(Bromo-acetic acid 3-(2,6-dioxo-1,3-dipropyl-2,3,6,...)
Affinity DataKd:  0.710nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039676BDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.710nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039680BDBM50039680(8-(2,5-Dioxo-2,5-dihydro-pyrrol-1-ylmethyl)-1,3-di...)
Affinity DataKd:  0.730nMAssay Description:Binding of [3H]-CPX to A1 adenosine receptor of DDT1 MF-2 (DDT) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039688BDBM50039688(4-[2-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  0.740nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080550BDBM50080550((2-amino-4,5-dimethylthien-3-yl)-[3-(trifluorometh...)
Affinity DataKd:  0.75nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039689BDBM50039689(3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKd:  0.790nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50023398BDBM50023398((4-{3-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82558BDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataKd:  0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095603BDBM50095603(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.810nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039678BDBM50039678(8-cyclopentyl-1,3-di[3-(4-fluorosulfonylphenylcarb...)
Affinity DataKd:  0.820nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039691BDBM50039691(3-[3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  0.860nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253928BDBM50253928((2-amino-4-((4-(4-(trifluoromethyl)phenyl)piperazi...)
Affinity DataKd:  1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253925BDBM50253925((2-amino-4-((4-p-tolylpiperazin-1-yl)methyl)thioph...)
Affinity DataKd:  1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253891BDBM50253891((2-amino-4-((4-(4-fluorophenyl)piperazin-1-yl)meth...)
Affinity DataKd:  1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253889BDBM50253889((2-amino-4-((4-phenylpiperazin-1-yl)methyl)thiophe...)
Affinity DataKd:  1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253308BDBM50253308((2-amino-4-((4-(pyrimidin-2-yl)piperazin-1-yl)meth...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039682BDBM50039682(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039697BDBM50039697(Bromo-acetic acid 2-(8-cyclopentyl-2,6-dioxo-1-pro...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253926BDBM50253926((2-amino-4-((4-(benzo[d][1,3]dioxol-5-yl)piperazin...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039685BDBM50039685(3-[2-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253927BDBM50253927(4-(4-((5-amino-4-(4-chlorobenzoyl)thiophen-3-yl)me...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253892BDBM50253892((2-amino-4-((4-(4-chlorophenyl)piperazin-1-yl)meth...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253890BDBM50253890((2-amino-4-((4-benzylpiperazin-1-yl)methyl)thiophe...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253888BDBM50253888((2-amino-4-((4-cyclohexylpiperazin-1-yl)methyl)thi...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080550BDBM50080550((2-amino-4,5-dimethylthien-3-yl)-[3-(trifluorometh...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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