Compile Data Set for Download or QSAR
Report error Found 319 of ki data for polymerid = 402,50003604,50004441,50004442,50004443
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50358609(CHEMBL1921858)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50229378((R)-N-(1-(3-(4-cyanophenyl)H-imidazo[1,2-a]pyridin...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]IP-10 from CXCR3 receptor expressed in human PBMC in RPMI-1640 buffer supplemented with 0.5% BSAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372007(CHEMBL257017)
Affinity DataKi:  3nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227864(1-(1-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  3nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50337250((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataKi:  3.16nMAssay Description:Displacement of [125I]CXCL10 from human CXCR3 expressed in HEK293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372000(CHEMBL256851)
Affinity DataKi:  4nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372006(CHEMBL256850)
Affinity DataKi:  5nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50227866(1-(8-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372008(CHEMBL444542)
Affinity DataKi:  6nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50227864(1-(1-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372005(CHEMBL429598)
Affinity DataKi:  6nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227866(1-(8-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  7nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372011(CHEMBL271847)
Affinity DataKi:  7nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227863(1-(1-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  9nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227863(1-(1-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  9nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50310502((R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydropyri...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]CXCL10 from CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227861(1-(3-fluoro-5-(trifluoromethyl)phenyl)-3-(1-((9-pi...)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227867(1-(1-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  11nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372015(CHEMBL402514)
Affinity DataKi:  15nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198419(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  16nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50301329(5-chloro-6-(4-((2S)-1-(4-chlorobenzyl)-2-methylpip...)
Affinity DataKi:  16nMAssay Description:Displacement of 125I-IP10 from recombinant human CXCR3 receptor expressed in Ba/F3 cell membrane after 1 to 4 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198419(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  16nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372012(CHEMBL404028)
Affinity DataKi:  18nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227865(1-(3-fluoro-5-(trifluoromethyl)phenyl)-3-(1-((8-pi...)
Affinity DataKi:  18nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372009(CHEMBL271636)
Affinity DataKi:  20nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227862(1-(1-((8-(cyclopropanecarbonyl)-8-aza-bicyclo[3.2....)
Affinity DataKi:  20nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372002(CHEMBL256188)
Affinity DataKi:  21nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372001(CHEMBL257018)
Affinity DataKi:  24nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372010(CHEMBL402245)
Affinity DataKi:  25nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50225715(3-(3,5-bis(trifluoromethyl)phenyl)-1-(1-(((1R,5S)-...)
Affinity DataKi:  26nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198392(1-(3,5-bis(trifluoromethyl)phenyl)-3-(1-(((1R,5S)-...)
Affinity DataKi:  26nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50372013(CHEMBL256190)
Affinity DataKi:  26nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227869(1-[1-(8-acetyl-8-aza-bicyclo[3.2.1]oct-2-en-3-ylme...)
Affinity DataKi:  27nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198395(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-...)
Affinity DataKi:  28nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50227873(1-(3-fluoro-5-(trifluoromethyl)phenyl)-3-(1-((8-is...)
Affinity DataKi:  28nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198405(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  29nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198390(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  31nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50301330(5-chloro-6-(4-((2S)-1-(4-chlorobenzyl)-2-methylpip...)
Affinity DataKi:  32nMAssay Description:Displacement of 125I-IP10 from recombinant human CXCR3 receptor expressed in Ba/F3 cell membrane after 1 to 4 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50227867(1-(1-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  33nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50301351(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-yl)pi...)
Affinity DataKi:  35nMAssay Description:Displacement of 125I-IP10 from recombinant human CXCR3 receptor expressed in Ba/F3 cell membrane after 1 to 4 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198415(1-(3,5-bis(trifluoromethyl)phenyl)-3-(1-(cycloocte...)
Affinity DataKi:  36nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50227863(1-(1-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)...)
Affinity DataKi:  38nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198389(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  39nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50399980(CHEMBL2181467)
Affinity DataKi:  39.8nMAssay Description:Displacement of [125I]CXCL10 from CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50211114((-)-(R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydro...)
Affinity DataKi:  39.8nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198418(1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(3,5-di...)
Affinity DataKi:  41nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198408(1-(5-(2-chlorophenyl)thiophen-2-yl)-3-(1-(((1R,5S)...)
Affinity DataKi:  46nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50198391(1-(1-(cyclooctenylmethyl)piperidin-4-yl)-3-(3-fluo...)
Affinity DataKi:  47nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
National Heart and Lung Institute

Curated by ChEMBL
LigandPNGBDBM50399981(CHEMBL2181450)
Affinity DataKi:  50.1nMAssay Description:Displacement of [125I]CXCL10 from CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50227861(1-(3-fluoro-5-(trifluoromethyl)phenyl)-3-(1-((9-pi...)
Affinity DataKi:  57nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
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