TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in absence of L-glutamic acid.More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in presence of 20 uM L-glutamic acidMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 6.60E+3nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in absence of L-glutamic acid in mammalian cellsMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.20E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.80E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in presence of 20 uM L-glutamic acid in mammalian cellsMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 4.60E+4nMAssay Description:Activity against human EAAT3 transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 4.90E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 5.10E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 5.20E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 6.60E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in absence of L-glutamic acid.More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 8.00E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 8.10E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 9.80E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+5nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >4.00E+5nMAssay Description:Activity against human EAAT3 transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.30E+5nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in presence of 20 uM L-glutamic acid.More data for this Ligand-Target Pair