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Report error Found 2081 Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein'
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50473322(CHEMBL302452)
Affinity DataKd:  3.20E+4nMAssay Description:Binding affinity towards 23-nt RNA oligonucleotide from the 5'-untranslated region of the cholestery ester transfer protein (CETP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50128131(SC-795 | 3-{[3-(4-Chloro-3-ethyl-phenoxy)-phenyl]-...)
Affinity DataIC50: 0.770nMAssay Description:Compound was tested in vitro for inhibitory activity against recombinant human cholesteryl ester transfer protein in buffer with <1 nM [CETP] for 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50392514(CHEMBL2152167)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant CETP using [3H]cholesterol ester/HDL as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50516404(CHEMBL4439823)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]CE/HDL transfer incubated for 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Rabbit)
Al-Zaytoonah Private University of Jordan

Curated by ChEMBL
LigandPNGBDBM50118064(1,1,1-trifluoro-3-((3-fluorophenyl)(3-(3-(trifluor...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50178701(CHEMBL3814374)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]cholesteryl ester transfer from [3H]CE-HDL to biotinylated LDL by scintillation pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254040(US9493430, 593)
Affinity DataIC50: 1.5nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50178698(CHEMBL3813720)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]cholesteryl ester transfer from [3H]CE-HDL to biotinylated LDL by scintillation pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254048(US9493430, 618)
Affinity DataIC50: 1.60nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50178699(CHEMBL3813836)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]cholesteryl ester transfer from [3H]CE-HDL to biotinylated LDL by scintillation pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254050(US9493430, 631)
Affinity DataIC50: 1.90nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254058(US9493430, 684)
Affinity DataIC50: 1.90nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50392527(CHEMBL2152180)
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant CETP using [3H]cholesterol ester/HDL as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50516410(CHEMBL4574163)
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]CE/HDL transfer incubated for 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254054(US9493430, 661)
Affinity DataIC50: 2.5nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50178702(CHEMBL3814963)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]cholesteryl ester transfer from [3H]CE-HDL to biotinylated LDL by scintillation pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50178700(CHEMBL3814418)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]cholesteryl ester transfer from [3H]CE-HDL to biotinylated LDL by scintillation pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234607(US9353101, 3)
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234610(US9353101, 6)
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234611(US9353101, 7)
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50128164(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-chlo...)
Affinity DataIC50: 3nMAssay Description:Inhibition of CETP-mediated transfer of [3H]cholesteryl ester from HDL donar particles to LDL acceptor particles in presence of bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50128164(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-chlo...)
Affinity DataIC50: 3nMAssay Description:Inhibition of CETP-mediated transfer of [3H]cholesteryl ester from HDL donar particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50312718(torcetrapib | CHEMBL479527)
Affinity DataIC50: 3nMAssay Description:Inhibition of human plasma CETP assessed as [3H]cholesterol ester transfer after 18 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholesteryl ester transfer protein(Rabbit)
Al-Zaytoonah Private University of Jordan

Curated by ChEMBL
LigandPNGBDBM50128137(3-{[3-(3-Ethyl-phenoxy)-phenyl]-[3-(1,1,2,2-tetraf...)
Affinity DataIC50: 3nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50094519((R)-3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-phe...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human CETP by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50392530(CHEMBL2152183)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant CETP using [3H]cholesterol ester/HDL as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50516398(CHEMBL4457286)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]CE/HDL transfer incubated for 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254034(US9493430, 574)
Affinity DataIC50: 3.90nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Rabbit)
Al-Zaytoonah Private University of Jordan

Curated by ChEMBL
LigandPNGBDBM50128131(SC-795 | 3-{[3-(4-Chloro-3-ethyl-phenoxy)-phenyl]-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234621(US9353101, 17)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234632(US9353101, 28)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234635(US9353101, 31)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234661(US9353101, 57)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234664(US9353101, 60)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254055(US9493430, 668)
Affinity DataIC50: 5nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50392513(CHEMBL2152166)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant CETP using [3H]cholesterol ester/HDL as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50516405(CHEMBL4552555)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]CE/HDL transfer incubated for 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50516406(CHEMBL4469874)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]CE/HDL transfer incubated for 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254037(US9493430, 584)
Affinity DataIC50: 5.30nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254030(US9493430, 557)
Affinity DataIC50: 5.40nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254028(US9493430, 554)
Affinity DataIC50: 5.80nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254066(US9493430, 756)
Affinity DataIC50: 5.90nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM192305(US9187450, 51)
Affinity DataIC50: 6nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and 5,5'-d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM192306(US9187450, 52)
Affinity DataIC50: 6nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and 5,5'-d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM234666(US9353101, 62)
Affinity DataIC50: 6nMpH: 7.4 T: 2°CAssay Description:Radiolabeled donor particles are generated by first combining 100 μl of 200 μM butylated hydroxyl toluene in CHCl3, 216 μL of 21.57 mM DOPC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50392504(CHEMBL2152158)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant CETP using [3H]cholesterol ester/HDL as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50392512(CHEMBL2152165)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant CETP using [3H]cholesterol ester/HDL as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50392528(CHEMBL2152181)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant CETP using [3H]cholesterol ester/HDL as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM50516400(CHEMBL4439856)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant CETP assessed as reduction in [3H]CE/HDL transfer incubated for 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Johann Wolfgang Goethe-Universit£T Frankfurt/Main

Curated by ChEMBL
LigandPNGBDBM254060(US9493430, 695)
Affinity DataIC50: 6.40nMAssay Description:As a protein source for cholesteryl ester transfer, plasma from healthy persons was used, and as a cholesteryl ester receptor, LDL from healthy perso...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent

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