Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 2743
TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378837BDBM378837(US10266528, Compound 14)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378836BDBM378836(US10266528, Compound 11)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378835BDBM378835(US10266528, Compound 19)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378834BDBM378834(US10266528, Compound 12 | US10266528, Compound 13)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378841BDBM378841(US10266528, Compound 16)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378840BDBM378840(US10266528, Compound 17)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378839BDBM378839(US10266528, Compound 23)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378838BDBM378838(US10266528, Compound 1)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378844BDBM378844(US10266528, Compound 21)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378843BDBM378843(US10266528, Compound 18)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378842BDBM378842(US10266528, Compound 2)
Affinity DataIC50: 10nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378851BDBM378851(US10266528, Compound 6)
Affinity DataIC50: 55nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378834BDBM378834(US10266528, Compound 12 | US10266528, Compound 13)
Affinity DataIC50: 55nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378845BDBM378845(US10266528, Compound 15)
Affinity DataIC50: 55nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378849BDBM378849(US10266528, Compound 22)
Affinity DataIC50: 55nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378848BDBM378848(US10266528, Compound 5)
Affinity DataIC50: 55nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378847BDBM378847(US10266528, Compound 4)
Affinity DataIC50: 55nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378846BDBM378846(US10266528, Compound 3)
Affinity DataIC50: 55nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378853BDBM378853(US10266528, Compound 7)
Affinity DataIC50: 550nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378852BDBM378852(US10266528, Compound 20)
Affinity DataIC50: 550nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378856BDBM378856(US10266528, Compound 8)
Affinity DataIC50: 1.00E+3nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378855BDBM378855(US10266528, Compound 9)
Affinity DataIC50: 1.00E+3nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 378854BDBM378854(US10266528, Compound 10)
Affinity DataIC50: 1.00E+3nMAssay Description:Briefly, 2.5× stocks of full-length human BTK (08-080) from CarnaBio USA, Inc., Natick, Mass., 1.6×ATP and appropriate kinKDR peptide substrate (FITC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent