Compile Data Set for Download or QSAR
Report error Found 491 Enz. Inhib. hit(s) with all data for entry = 8731
LigandChemical structure of BindingDB Monomer ID 415317BDBM415317(US10428044, Example 426 | 3-{[2-(hydroxymethyl)phe...)
Affinity DataIC50: 2.58nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415374BDBM415374(US10428044, Example 487 | 3-{[5-fluoro-2-(hydroxym...)
Affinity DataIC50: 3.35nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415373BDBM415373(US10428044, Example 486 | 3-{[3-fluoro-2-(hydroxym...)
Affinity DataIC50: 3.45nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415303BDBM415303(US10428044, Example 410 | Intermediate 1-2-69)
Affinity DataIC50: 3.55nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415283BDBM415283(US10428044, Example 390 | 1-(1-methyl-1H-pyrazol-4...)
Affinity DataIC50: 3.96nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414909BDBM414909(US10428044, Example 7 | US10428044, Example 18 | U...)
Affinity DataIC50: 4.04nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415365BDBM415365(US10428044, Example 478 | 1-benzyl-N-{4-[6,6-dimet...)
Affinity DataIC50: 4.23nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415336BDBM415336(US10428044, Example 449 | 1-benzyl-N-{4-[4-oxo-3-(...)
Affinity DataIC50: 4.38nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415357BDBM415357(US10428044, Example 470 | N-{4-[4′-oxo-3R...)
Affinity DataIC50: 4.49nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415284BDBM415284(US10428044, Example 391 | 1-{4-[6,6-dimethyl-4-oxo...)
Affinity DataIC50: 4.52nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415331BDBM415331(US10428044, Example 444 | 2-{[(2-aminopyridin-4-yl...)
Affinity DataIC50: 4.61nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415353BDBM415353(US10428044, Example 466 | rel-(R,S)-2-fluoro-N-{4-...)
Affinity DataIC50: 5.03nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415359BDBM415359(US10428044, Example 472 | 1-tert-butyl-N-{4-[6,6-d...)
Affinity DataIC50: 5.04nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415330BDBM415330(US10428044, Example 443 | 6-(chloromethyl)-3-(phen...)
Affinity DataIC50: 5.05nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415366BDBM415366(US10428044, Example 479 | N-{4-[6,6-dimethyl-4-oxo...)
Affinity DataIC50: 5.09nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414909BDBM414909(US10428044, Example 7 | US10428044, Example 18 | U...)
Affinity DataIC50: 5.09nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415379BDBM415379(US10428044, Example 492 | N-{4-[4-oxo-3-(phenylami...)
Affinity DataIC50: 5.28nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414932BDBM414932(3-[(3,5-difluorophenyl)amino]-6,6-dimethyl-2-(pyri...)
Affinity DataIC50: 5.55nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414909BDBM414909(US10428044, Example 7 | US10428044, Example 18 | U...)
Affinity DataIC50: 5.57nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414931BDBM414931(2-(3-fluoropyridin-4-yl)-6,6-dimethyl-3-(phenylami...)
Affinity DataIC50: 5.69nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415372BDBM415372(US10428044, Example 485 | 3-{[4-fluoro-2-(hydroxym...)
Affinity DataIC50: 5.84nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414929BDBM414929(6-ethyl-3-(phenylamino)-2-(pyridin-4-yl)-1,5,6,7-t...)
Affinity DataIC50: 5.93nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415391BDBM415391(US10428044, Example 504 | N-{4-[6,6-dimethyl-4-oxo...)
Affinity DataIC50: 6.14nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414930BDBM414930(6-(2-methylpropyl)-3-(phenylamino)-2-(pyridin-4-yl...)
Affinity DataIC50: 6.17nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415244BDBM415244(US10428044, Example 351 | 2-[(1-methyl-1H-pyrazol-...)
Affinity DataIC50: 6.22nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415337BDBM415337(US10428044, Example 450 | 1-(4-methoxybenzyl)-N-{4...)
Affinity DataIC50: 6.24nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414900BDBM414900(6,6-dimethyl-3-(phenylamino)-2-(pyridin-4- yl)-1,5...)
Affinity DataIC50: 6.25nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415367BDBM415367(US10428044, Example 480 | N-{4-[6,6-dimethyl-4-oxo...)
Affinity DataIC50: 6.30nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415152BDBM415152(US10428044, Example 254 | (S,R) N-{4-[6,6-dimethyl...)
Affinity DataIC50: 6.34nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415108BDBM415108(2′-(3-fluoropyridin-4-yl)-3′-(phenylam...)
Affinity DataIC50: 6.39nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415301BDBM415301(US10428044, Example 408 | Intermediate 1-2-68)
Affinity DataIC50: 6.42nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415248BDBM415248(US10428044, Example 355 | 2-[(5-methyl-1,3-oxazol-...)
Affinity DataIC50: 6.45nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415383BDBM415383(US10428044, Example 496 | 2-[(4-methyl-1,3-thiazol...)
Affinity DataIC50: 6.46nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415243BDBM415243(US10428044, Example 350 | 2-[(3-methyl-1,2-oxazol-...)
Affinity DataIC50: 6.53nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 414915BDBM414915(3′-(phenylamino)-2′-(pyridin-4-yl)-1&#...)
Affinity DataIC50: 6.55nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415247BDBM415247(US10428044, Example 354 | 2-[(5-methyl-1,2-oxazol-...)
Affinity DataIC50: 6.57nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415364BDBM415364(US10428044, Example 477 | N-{4-[6,6-dimethyl-4-oxo...)
Affinity DataIC50: 6.62nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415167BDBM415167(US10428044, Example 272 | N-{4-[6,6-dimethyl-4-oxo...)
Affinity DataIC50: 6.63nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415245BDBM415245(US10428044, Example 352 | 2-(furan-2-ylmethoxy)-N-...)
Affinity DataIC50: 6.68nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415304BDBM415304(US10428044, Example 411 | Intermediate 1-2-70)
Affinity DataIC50: 6.86nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415348BDBM415348(US10428044, Example 461 | N-{4-[6-(fluoromethyl)-4...)
Affinity DataIC50: 6.88nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415329BDBM415329(US10428044, Example 442 | Intermediate 1-1-32)
Affinity DataIC50: 6.97nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415235BDBM415235(US10428044, Example 342 | 2-[(4-methoxybenzyl)oxy]...)
Affinity DataIC50: 7.12nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415352BDBM415352(US10428044, Example 465 | N-{4-[6,6-dimethyl-4-oxo...)
Affinity DataIC50: 7.19nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415233BDBM415233(US10428044, Example 340 | 2-(benzyloxy)-N-{4-[4-ox...)
Affinity DataIC50: 7.25nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415107BDBM415107(Intermediate 1-2-37 | US10428044, Example 207)
Affinity DataIC50: 7.32nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415341BDBM415341(US10428044, Example 454 | 1-methyl-N-{4-[4-oxo-3-(...)
Affinity DataIC50: 7.33nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415226BDBM415226(US10428044, Example 333 | 2-butoxy-N-{4-[4-oxo-3-(...)
Affinity DataIC50: 7.33nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415149BDBM415149(US10428044, Example 249 | rel-(R,S/S,R)-2-fluoro-N...)
Affinity DataIC50: 7.55nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415166BDBM415166(US10428044, Example 271 | N-{4-[4-oxo-3-(phenylami...)
Affinity DataIC50: 7.64nMAssay Description:In a typical assay 11 different concentrations of each compound (0.1 nM, 0.33 nM, 1.1 nM, 3.8 nM, 13 nM, 44 nM, 0.15 μM, 0.51 μM, 1.7 μ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
US Patent

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