Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 11661
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637599BDBM637599(US20230382915, Example 33)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637568BDBM637568(US20230382915, Example 1)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637569BDBM637569(US20230382915, Example 2 | US20230382915, Example ...)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637597BDBM637597(US20230382915, Example 31)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637598BDBM637598(US20230382915, Example 32)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637598BDBM637598(US20230382915, Example 32)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637599BDBM637599(US20230382915, Example 33)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637571BDBM637571(US20230382915, Example 4)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637572BDBM637572(US20230382915, Example 5)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637569BDBM637569(US20230382915, Example 2 | US20230382915, Example ...)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637570BDBM637570(US20230382915, Example 3)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637570BDBM637570(US20230382915, Example 3)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637571BDBM637571(US20230382915, Example 4)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637591BDBM637591(US20230382915, Example 24)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637592BDBM637592(US20230382915, Example 25)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637590BDBM637590(US20230382915, Example 23 | US20230382915, Example...)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637589BDBM637589(US20230382915, Example 22)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637590BDBM637590(US20230382915, Example 23 | US20230382915, Example...)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637595BDBM637595(US20230382915, Example 29)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637597BDBM637597(US20230382915, Example 31)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637590BDBM637590(US20230382915, Example 23 | US20230382915, Example...)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637569BDBM637569(US20230382915, Example 2 | US20230382915, Example ...)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637569BDBM637569(US20230382915, Example 2 | US20230382915, Example ...)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637583BDBM637583(US20230382915, Example 16)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637584BDBM637584(US20230382915, Example 17)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637584BDBM637584(US20230382915, Example 17)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637581BDBM637581(US20230382915, Example 14)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637582BDBM637582(US20230382915, Example 15)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637582BDBM637582(US20230382915, Example 15)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637583BDBM637583(US20230382915, Example 16)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637587BDBM637587(US20230382915, Example 20)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637588BDBM637588(US20230382915, Example 21)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637588BDBM637588(US20230382915, Example 21)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637585BDBM637585(US20230382915, Example 18)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637586BDBM637586(US20230382915, Example 19)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637575BDBM637575(US20230382915, Example 8)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637576BDBM637576(US20230382915, Example 9)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637577BDBM637577(US20230382915, Example 10)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637573BDBM637573(US20230382915, Example 6)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637574BDBM637574(US20230382915, Example 7)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637575BDBM637575(US20230382915, Example 8)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637579BDBM637579(US20230382915, Example 12)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637580BDBM637580(US20230382915, Example 13)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637581BDBM637581(US20230382915, Example 14)
Affinity DataIC50: 100nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637577BDBM637577(US20230382915, Example 10)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637578BDBM637578(US20230382915, Example 11)
Affinity DataIC50: 100nMAssay Description:Activity of PERK kinase was determined spectroscopically using a coupled pyruvate kinase/lactate dehydrogenase assay that continuously monitors the A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637592BDBM637592(US20230382915, Example 25)
Affinity DataIC50: 300nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637590BDBM637590(US20230382915, Example 23 | US20230382915, Example...)
Affinity DataIC50: 300nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637574BDBM637574(US20230382915, Example 7)
Affinity DataIC50: 300nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

TargeteIF-2-alpha kinase GCN2(Human)
Deciphera Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 637580BDBM637580(US20230382915, Example 13)
Affinity DataIC50: 300nMAssay Description:Activity of GCN2 kinase was determined using a TR-FRET kinase activity assay (e.g. Riddle et al. Analytical Biochemistry (2006) 356(1) 108-116). Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
US Patent

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