Compile Data Set for Download or QSAR
Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 12743
LigandChemical structure of BindingDB Monomer ID 724688BDBM724688(N-((1r,4r)-4-(4-acet- ylpiperazin-1-yl)- cyclohexy...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724716BDBM724716(N-((1r,4r)-4-(4-acet- ylpiperazin-1-yl)- cyclohexy...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724724BDBM724724(N-((1r,4r)-4-(3- methoxyazetidin-1- yl)cyclohexyl)...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724691BDBM724691(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (4-(2,2...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724689BDBM724689(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (4-isop...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724721BDBM724721(N-((1r,4r)-4-(3- (difluoromethoxy)- azetidin-1-yl)...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724688BDBM724688(N-((1r,4r)-4-(4-acet- ylpiperazin-1-yl)- cyclohexy...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724720BDBM724720(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (3-(dif...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724689BDBM724689(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (4-isop...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724721BDBM724721(N-((1r,4r)-4-(3- (difluoromethoxy)- azetidin-1-yl)...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724711BDBM724711(3-methyl-N-((1r,4r)- 4-morpholinocyclo- hexyl)-1-n...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724710BDBM724710(N-((1r,4r)-4-(4-iso- propylpiperazin-1- yl)cyclohe...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724711BDBM724711(3-methyl-N-((1r,4r)- 4-morpholinocyclo- hexyl)-1-n...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724709BDBM724709(N-((1r,4r)-4-(3,3- difluoroazetidin-1- yl)cyclohex...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724710BDBM724710(N-((1r,4r)-4-(4-iso- propylpiperazin-1- yl)cyclohe...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724709BDBM724709(N-((1r,4r)-4-(3,3- difluoroazetidin-1- yl)cyclohex...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724715BDBM724715(N-((1r,4r)-4-(3- cyanoazetidin-1-yl)- cyclohexyl)-...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724716BDBM724716(N-((1r,4r)-4-(4-acet- ylpiperazin-1-yl)- cyclohexy...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724715BDBM724715(N-((1r,4r)-4-(3- cyanoazetidin-1-yl)- cyclohexyl)-...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724703BDBM724703(N-((1r,4r)-4-(4-cyclo- propylpiperazin-1-yl)- cycl...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724703BDBM724703(N-((1r,4r)-4-(4-cyclo- propylpiperazin-1-yl)- cycl...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724675BDBM724675(N-((1r,4r)-4-(4-acetyl- piperazin-1-yl)cyclo- hexy...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724706BDBM724706(N-((1r,4r)-4-(3,3- difluoropyrrolidin-1- yl)cycloh...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724675BDBM724675(N-((1r,4r)-4-(4-acetyl- piperazin-1-yl)cyclo- hexy...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724705BDBM724705(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (3,3-di...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724706BDBM724706(N-((1r,4r)-4-(3,3- difluoropyrrolidin-1- yl)cycloh...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724705BDBM724705(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (3,3-di...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724696BDBM724696(N-((1r,4r)-4-(3,3- difluoroazetidin-1- yl)cyclohex...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724696BDBM724696(N-((1r,4r)-4-(3,3- difluoroazetidin-1- yl)cyclohex...)
Affinity DataIC50: 10nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724720BDBM724720(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (3-(dif...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724684BDBM724684(1-isobutyl-N-((1r,4r)- 4-(4-isopropylpiper- azin-1...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724685BDBM724685(N-((1r,4r)-4-(4-cyclo- propylpiperazin-1-yl)- cycl...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724691BDBM724691(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (4-(2,2...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724692BDBM724692(1-(4,4-difluorocyclo- hexyl)-3-methyl-N- ((1r,4r)-...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724690BDBM724690(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (4-(2,2...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724722BDBM724722(N-((1r,4r)-4-(3- cyanoazetidin-1-yl)- cyclohexyl)-...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724690BDBM724690(1-(4,4-difluorocyclo- hexyl)-N-((1r,4r)-4- (4-(2,2...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724722BDBM724722(N-((1r,4r)-4-(3- cyanoazetidin-1-yl)- cyclohexyl)-...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724712BDBM724712(N-((1r,3r)-3-(4-cyclo- propylpiperazin-1- yl)cyclo...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724678BDBM724678(1-(2-chlorophenyl)-N- ((1r,4r)-4-(3-(difluoro- met...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724678BDBM724678(1-(2-chlorophenyl)-N- ((1r,4r)-4-(3-(difluoro- met...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724708BDBM724708(N-((1r,3r)-3-(4-acet- ylpiperazin-1-yl)- cyclobuty...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724682BDBM724682(1-(4,4-difluorocyclo- hexyl)-N-(3-(3,3- difluoropy...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724714BDBM724714(3-methyl-N-(6- morpholinopyridin- 3-yl)-1-neopenty...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724683BDBM724683(N-((1r,4r)-4-(3,3- difluoroazetidin-1-yl)- cyclohe...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724682BDBM724682(1-(4,4-difluorocyclo- hexyl)-N-(3-(3,3- difluoropy...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724714BDBM724714(3-methyl-N-(6- morpholinopyridin- 3-yl)-1-neopenty...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724712BDBM724712(N-((1r,3r)-3-(4-cyclo- propylpiperazin-1- yl)cyclo...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724713BDBM724713(N-((1r,3r)-3-(4-cyclo- propylpiperazin-1- yl)cyclo...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 724704BDBM724704(3-methyl-N-((1r,3r)- 3-morpholinocyclo- butyl)-1-n...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

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