Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 13482
TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 50395554BDBM50395554(CHEMBL161792 | US20260076975, Compound 10)
Affinity DataEC50:  130nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798239BDBM798239(US20260076975, Compound 150)
Affinity DataEC50:  139nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798223BDBM798223(4-(5-(4-(2,3-dichlorophenyl)piperazin-1-yl)pentyl)...)
Affinity DataEC50:  220nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 50130293BDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataEC50:  460nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798221BDBM798221((E)-2-(4-(3-(3,4-dimethoxyphenyl)allyl)piperazin-1...)
Affinity DataEC50:  650nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798198BDBM798198(6-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)...)
Affinity DataEC50:  754nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798216BDBM798216((E)-5-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)pro...)
Affinity DataEC50:  918nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798207BDBM798207(7-(4-(4-(2-methyl-10H-benzo[b]thieno[2,3-e][1,4]di...)
Affinity DataEC50:  1.00E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798197BDBM798197(7-((5-(4-(2,3-dichlorophenyl)piperazin-1-yl)pentyl...)
Affinity DataEC50:  1.01E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798234BDBM798234(US20260076975, Compound 138)
Affinity DataEC50:  1.01E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798189BDBM798189(7-((5-(4-(2,3-dichlorophenyl)piperazin-1-yl)pentyl...)
Affinity DataEC50:  1.04E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798195BDBM798195(N-(4-(2,3-dichlorophenyl)cyclohexyl)-2-((2-oxo-1,2...)
Affinity DataEC50:  1.06E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798209BDBM798209(2-((2-(4-(3,5-bis(trifluoromethyl)phenyl)piperazin...)
Affinity DataEC50:  1.07E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798208BDBM798208(6-(4-(4-(benzo[d]thiazol-2-yl)piperazin-1-yl)butox...)
Affinity DataEC50:  1.14E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 63372BDBM63372(7-((4-(4-(2,3-dichlorophenyl)piperazin-1-yl)but-1-...)
Affinity DataEC50:  1.16E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798205BDBM798205(7-(4-(4-(benzo[d]thiazol-2-yl)piperazin-1-yl)butox...)
Affinity DataEC50:  1.17E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798192BDBM798192(7-((5-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl...)
Affinity DataEC50:  1.18E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798206BDBM798206(7-(3-(4-(benzo[d]thiazol-2-yl)piperazin-1-yl)propo...)
Affinity DataEC50:  1.18E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 50395582BDBM50395582(CHEMBL2165133 | UNC10000004 | US9156822, 25 | US20...)
Affinity DataEC50:  1.19E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798219BDBM798219(1-(2,3-dichlorophenyl)-4-(4-(5-methoxypyridin-3-yl...)
Affinity DataEC50:  1.19E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 50395555BDBM50395555(CHEMBL2165127 | US20260076975, Compound 5)
Affinity DataEC50:  1.20E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798213BDBM798213(US20260076975, Compound 58)
Affinity DataEC50:  1.20E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 312188BDBM312188(US9604944, 15b (Example 14) | 6-(4-(4-(2,3-Dichlor...)
Affinity DataEC50:  1.22E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798214BDBM798214((E)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)-4-(3,...)
Affinity DataEC50:  1.22E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798238BDBM798238(US20260076975, Compound 148)
Affinity DataEC50:  1.23E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798191BDBM798191(7-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)...)
Affinity DataEC50:  1.27E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798215BDBM798215((E)-1-(2,3-dichlorophenyl)-4-(3-(3,4-dimethoxyphen...)
Affinity DataEC50:  1.28E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798202BDBM798202(7-(2-(4-(benzo[d]thiazol-2-yl)piperazin-1-yl)ethox...)
Affinity DataEC50:  1.30E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798210BDBM798210(2-(((4-(2,3-dichlorophenyl)piperazin-1-yl)-2-oxoet...)
Affinity DataEC50:  1.31E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798204BDBM798204(7-(4-(4-(benzo[d]thiazol-2-yl)piperazin-1-yl)butox...)
Affinity DataEC50:  1.32E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798237BDBM798237(US20260076975, Compound 146)
Affinity DataEC50:  1.34E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798203BDBM798203(7-(2-(4-(benzothiazol-2-yl)piperazin-1-yl)ethoxy)q...)
Affinity DataEC50:  1.37E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798200BDBM798200(6-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propoxy...)
Affinity DataEC50:  1.54E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798201BDBM798201(6-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butoxy)...)
Affinity DataEC50:  2.28E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798226BDBM798226(ethyl 2-((4-(4-(2,3-dichlorophenyl)piperazin-1-yl)...)
Affinity DataEC50:  2.52E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798225BDBM798225(ethyl 2-((4-(4-(benzo[d]thiazol-2-yl)piperazin-1-y...)
Affinity DataEC50:  2.55E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798243BDBM798243(US20260076975, Compound 157)
Affinity DataEC50:  2.61E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798218BDBM798218(1-(2,3-dichlorophenyl)-4-(3-(5-methoxypyridin-3-yl...)
Affinity DataEC50:  2.72E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 50001786BDBM50001786(1-[2-[4-[5-chloro-1-(4-fluorophenyl)-indol-3-yl]-1...)
Affinity DataEC50:  2.80E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798220BDBM798220(1-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-(5-meth...)
Affinity DataEC50:  3.24E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798240BDBM798240(US20260076975, Compound 151)
Affinity DataEC50:  3.36E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798224BDBM798224(N-(2-(4-(5-chloro-2-methylphenyl)piperazin-1-yl)et...)
Affinity DataEC50:  3.46E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798212BDBM798212(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)-N-(3-(dim...)
Affinity DataEC50:  3.80E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798227BDBM798227(US20260076975, Compound 84)
Affinity DataEC50:  3.86E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798245BDBM798245(1-(6-(4-(2,3-dichlorophenyl)piperazine-1-carbonyl)...)
Affinity DataEC50:  4.25E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798248BDBM798248(N-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)-4-oxob...)
Affinity DataEC50:  4.39E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798211BDBM798211(N-(3-amino-4-methoxyphenyl)-2-(4-(2,3-dichlorophen...)
Affinity DataEC50:  4.65E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798217BDBM798217(4-(2,3-dichlorophenyl)-N-(3,4-dimethoxyphenethyl)p...)
Affinity DataEC50:  4.71E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 50395556BDBM50395556(CHEMBL2165125 | US20260076975, Compound 19)
Affinity DataEC50:  5.01E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetThiamine pyrophosphokinase 1(Human)
Shanghai Raising Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 798246BDBM798246(1-(6-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-3,4...)
Affinity DataEC50:  5.43E+3nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

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