Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 6053
TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106687BDBM106687(US8586571, 50)
Affinity DataIC50: 5nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106685BDBM106685(US8586571, 17)
Affinity DataIC50: 10nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106694BDBM106694(US8586571, 207)
Affinity DataIC50: 12nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106691BDBM106691(US8586571, 164)
Affinity DataIC50: 15nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106681BDBM106681(US8586571, 6)
Affinity DataIC50: 20nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106688BDBM106688(US8586571, 80)
Affinity DataIC50: 20nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106690BDBM106690(US8586571, 143)
Affinity DataIC50: 23nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106684BDBM106684(US8586571, 14)
Affinity DataIC50: 24nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106695BDBM106695(US8586571, 215)
Affinity DataIC50: 34nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106682BDBM106682(US8586571, 36)
Affinity DataIC50: 36nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106693BDBM106693(US8586571, 197)
Affinity DataIC50: 40nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106692BDBM106692(US8586571, 189)
Affinity DataIC50: 71nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106683BDBM106683(US8586571, 12)
Affinity DataIC50: 210nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106686BDBM106686(US8586571, 20)
Affinity DataIC50: 290nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent

TargetRetinol-binding protein 4(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 106689BDBM106689(US8586571, 121)
Affinity DataIC50: 790nMAssay Description:The action of the compound of the present invention to inhibit binding of RBP4 and retinol and TTR was evaluated using the Retinol-RBP4-TTR ELISA (hu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2014
Entry Details
US Patent