Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 6418
LigandChemical structure of BindingDB Monomer ID 20557BDBM20557(N-[4-({6-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl...)
Affinity DataIC50: 20nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128023BDBM128023(US8796328, C)
Affinity DataIC50: 35nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128033BDBM128033(US8796328, 10)
Affinity DataIC50: 54nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128022BDBM128022(US8802711, I | US8796328, B)
Affinity DataIC50: 55nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50264258BDBM50264258(US8796328, E | CHEMBL523605 | 1-(3-Methylpyridin-2...)
Affinity DataIC50: 100nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128024BDBM128024(US8796328, 1)
Affinity DataIC50: 104nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128032BDBM128032(US8796328, 9)
Affinity DataIC50: 109nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50321851BDBM50321851(CHEMBL1173240 | US8796328, D | (R)-8-{5-[3-Methyl-...)
Affinity DataIC50: 180nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128037BDBM128037(US8796328, 14)
Affinity DataIC50: 209nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128057BDBM128057(US8796328, 37)
Affinity DataIC50: 256nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128028BDBM128028(US8796328, 5)
Affinity DataIC50: 325nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128031BDBM128031(US8796328, 8)
Affinity DataIC50: 330nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128058BDBM128058(US8796328, 38)
Affinity DataIC50: 345nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128046BDBM128046(US8796328, 23)
Affinity DataIC50: 358nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128036BDBM128036(US8796328, 13)
Affinity DataIC50: 418nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128042BDBM128042(US8796328, 19)
Affinity DataIC50: 466nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128056BDBM128056(US8796328, 36)
Affinity DataIC50: 587nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128047BDBM128047(US8796328, 25)
Affinity DataIC50: 602nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128059BDBM128059(US8796328, 39)
Affinity DataIC50: 615nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128030BDBM128030(US8796328, 7)
Affinity DataIC50: 747nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128043BDBM128043(US8796328, 20)
Affinity DataIC50: 791nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128038BDBM128038(US8796328, 15)
Affinity DataIC50: 863nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128054BDBM128054(US8796328, 32)
Affinity DataIC50: 913nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128051BDBM128051(US8796328, 29)
Affinity DataIC50: 1.15E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128064BDBM128064(US8796328, 44)
Affinity DataIC50: 1.28E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128026BDBM128026(US8796328, 3)
Affinity DataIC50: 1.81E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128041BDBM128041(US8796328, 18)
Affinity DataIC50: 2.15E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128055BDBM128055(US8796328, 35)
Affinity DataIC50: 2.44E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128029BDBM128029(US8796328, 6)
Affinity DataIC50: 2.90E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128040BDBM128040(US8796328, 17)
Affinity DataIC50: 3.03E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128053BDBM128053(US8796328, 31)
Affinity DataIC50: 3.80E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128061BDBM128061(US8796328, 41)
Affinity DataIC50: 5.28E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128063BDBM128063(US8796328, 43)
Affinity DataIC50: 6.41E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128044BDBM128044(US8796328, 21)
Affinity DataIC50: 7.56E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128045BDBM128045(US8796328, 22)
Affinity DataIC50: 7.59E+3nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128060BDBM128060(US8796328, 40)
Affinity DataIC50: 1.01E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128027BDBM128027(US8796328, 4)
Affinity DataIC50: 1.65E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128049BDBM128049(US8796328, 27)
Affinity DataIC50: 2.25E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128039BDBM128039(US8796328, 16)
Affinity DataIC50: 2.28E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128050BDBM128050(US8796328, 28)
Affinity DataIC50: 2.95E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128062BDBM128062(US8796328, 42)
Affinity DataIC50: 3.28E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128048BDBM128048(US8796328, 26)
Affinity DataIC50: 3.75E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128052BDBM128052(US8796328, 30)
Affinity DataIC50: 3.75E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 128035BDBM128035(US8796328, 12)
Affinity DataIC50: 3.75E+4nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
US Patent