Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 6758
TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151169BDBM151169(US8987286, 15.3)
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151167BDBM151167(US8987286, 15.1)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151168BDBM151168(US8987286, 15.2)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151153BDBM151153(US8987286, 6.6)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151170BDBM151170(US8987286, 15.4)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151142BDBM151142(US8987286, 4.12)
Affinity DataIC50: 14nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151166BDBM151166(US8987286, 15)
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151150BDBM151150(US8987286, 6.3)
Affinity DataIC50: 16nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151139BDBM151139(US8987286, 4.9)
Affinity DataIC50: 16nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151141BDBM151141(US8987286, 4.11)
Affinity DataIC50: 17nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151151BDBM151151(US8987286, 6.4)
Affinity DataIC50: 18nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151154BDBM151154(US8987286, 6.7)
Affinity DataIC50: 19nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151140BDBM151140(US8987286, 4.10)
Affinity DataIC50: 21nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151143BDBM151143(US8987286, 4.13)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151137BDBM151137(US8987286, 4.7)
Affinity DataIC50: 25nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151171BDBM151171(US8987286, 15.5)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151152BDBM151152(US8987286, 6.5)
Affinity DataIC50: 31nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151135BDBM151135(US8987286, 4.5)
Affinity DataIC50: 35nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151148BDBM151148(US8987286, 6.1)
Affinity DataIC50: 41nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151134BDBM151134(US8987286, 4.4)
Affinity DataIC50: 43nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151162BDBM151162(US8987286, 9)
Affinity DataIC50: 49nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151131BDBM151131(US8987286, 4.1)
Affinity DataIC50: 59nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151147BDBM151147(US8987286, 6)
Affinity DataIC50: 67nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151133BDBM151133(US8987286, 4.3)
Affinity DataIC50: 87nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151127BDBM151127(US8987286, 1)
Affinity DataIC50: 93nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151149BDBM151149(US8987286, 6.2)
Affinity DataIC50: 97nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151164BDBM151164(US8987286, 11)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151144BDBM151144(US8987286, 5)
Affinity DataIC50: 110nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151138BDBM151138(US8987286, 4.8)
Affinity DataIC50: 111nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151145BDBM151145(US8987286, 5.1)
Affinity DataIC50: 120nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151146BDBM151146(US8987286, 5.2)
Affinity DataIC50: 130nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151130BDBM151130(US8987286, 4)
Affinity DataIC50: 140nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151161BDBM151161(US8987286, 8.5)
Affinity DataIC50: 160nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151157BDBM151157(US8987286, 8.1)
Affinity DataIC50: 170nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151132BDBM151132(US8987286, 4.2)
Affinity DataIC50: 229nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151155BDBM151155(US8987286, 7)
Affinity DataIC50: 320nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151136BDBM151136(US8987286, 4.6)
Affinity DataIC50: 458nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151128BDBM151128(US8987286, 2)
Affinity DataIC50: 528nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151165BDBM151165(US8987286, 14)
Affinity DataIC50: 580nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151159BDBM151159(US8987286, 8.3)
Affinity DataIC50: 720nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151163BDBM151163(US8987286, 10)
Affinity DataIC50: 740nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151129BDBM151129(US8987286, 3)
Affinity DataIC50: 2.63E+3nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151158BDBM151158(US8987286, 8.2)
Affinity DataIC50: 5.60E+3nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151156BDBM151156(US8987286, 8)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent

TargetRAC-alpha serine/threonine-protein kinase(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 151160BDBM151160(US8987286, 8.4)
Affinity DataIC50: 1.70E+4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nl of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
US Patent