Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 6874
TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155349BDBM155349(US9006268, 21)
Affinity DataIC50: 0.700nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155348BDBM155348(US9006268, 19)
Affinity DataIC50: 0.780nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155351BDBM155351(US9006268, 23)
Affinity DataIC50: 2.40nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155350BDBM155350(US9006268, 22)
Affinity DataIC50: 4.40nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155354BDBM155354(US9006268, 10)
Affinity DataIC50: 8nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155345BDBM155345(US9006268, 3)
Affinity DataIC50: 12nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155352BDBM155352(US9006268, 24)
Affinity DataIC50: 32nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155353BDBM155353(US9006268, 25)
Affinity DataIC50: 35nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155347BDBM155347(US9006268, 11)
Affinity DataIC50: 114nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent

TargetLysosomal Pro-X carboxypeptidase(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 155346BDBM155346(US9006268, 9)
Affinity DataIC50: 554nMpH: 5.5Assay Description:The assay was run in a 384-well microtiter plate at 37 ° C. with a total volume of 50 uL. Final assay concentrations were 0.13 nM human PrCP (CHO) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
US Patent