Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 6940
TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 47952BDBM47952(MLS000588669 | N-[3-(4-methylphenyl)sulfonyl-1-pro...)
Affinity DataIC50: 500nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 54915BDBM54915(cid_1930124 | N-[1-butyl-3-(4-methylphenyl)sulfony...)
Affinity DataIC50: 500nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 30831BDBM30831(MLS000055622 | N-(1-butyl-3-cyano-2-pyrrolo[3,2-b]...)
Affinity DataIC50: 760nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 160656BDBM160656(US9045483, 9)
Affinity DataIC50: 1.10E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 32062BDBM32062(SMR000060333 | MLS000054842 | N-(1-butyl-3-cyanopy...)
Affinity DataIC50: 3.60E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 160655BDBM160655(US9045483, 8)
Affinity DataIC50: 4.50E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 160657BDBM160657(US9045483, 10)
Affinity DataIC50: 5.70E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 37640BDBM37640(N-(1-butyl-3-cyano-pyrrolo[3,2-b]quinoxalin-2-yl)e...)
Affinity DataIC50: 8.30E+3nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 30722BDBM30722(cid_658797 | SMR000039762 | MLS000068755 | N-(1-bu...)
Affinity DataIC50: 2.00E+4nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 43094BDBM43094(2-chloranyl-N-[3-cyano-1-(phenylmethyl)pyrrolo[3,2...)
Affinity DataIC50: 2.50E+4nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 160653BDBM160653(US9045483, 6)
Affinity DataIC50: 6.40E+4nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 160654BDBM160654(US9045483, 7)
Affinity DataIC50: 9.80E+4nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSUMO-activating enzyme subunit 1/2(Human)
City of Hope

US Patent
LigandChemical structure of BindingDB Monomer ID 160658BDBM160658(US9045483, 11)
Affinity DataIC50: 1.00E+5nMAssay Description:Through the Molecular Library Probe Production Center Network (MLPCN), at least 300,000 compounds were screened using a TR-FRET method, an ALPHASCREE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent