Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 7267
TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185661BDBM185661(US9161922, Table 4, Compound 3)
Affinity DataIC50: 500nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185660BDBM185660(US9161922, Table 4, Compound 2)
Affinity DataIC50: 500nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185659BDBM185659(US9161922, Table 4, Compound 1)
Affinity DataIC50: 500nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185662BDBM185662(US9161922, Table 4, Compound 5 | US9161922, Table ...)
Affinity DataIC50: 1.10E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185662BDBM185662(US9161922, Table 4, Compound 5 | US9161922, Table ...)
Affinity DataIC50: 1.20E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185644BDBM185644(US9161922, Table 1, Compound 10)
Affinity DataIC50: 2.00E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185655BDBM185655(US9161922, Table 2, Compound 10)
Affinity DataIC50: 2.00E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185646BDBM185646(US9161922, Table 2, Compound 2 | US9161922, Table ...)
Affinity DataIC50: 2.90E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185651BDBM185651(US9161922, Table 2, Compound 6)
Affinity DataIC50: 3.60E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185652BDBM185652(US9161922, Table 2, Compound 7)
Affinity DataIC50: 4.60E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetHistamine oxidase(Arthrobacter globiformis)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185658BDBM185658(US9161922, Table 3, Compound 3)
Affinity DataIC50: 7.00E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185649BDBM185649(US9161922, Table 2, Compound 4)
Affinity DataIC50: 8.40E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185641BDBM185641(US9161922, Table 1, Compound 7)
Affinity DataIC50: 9.00E+3nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185638BDBM185638(US9161922, Table 1, Compound 4)
Affinity DataIC50: 1.00E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185646BDBM185646(US9161922, Table 2, Compound 2 | US9161922, Table ...)
Affinity DataIC50: 1.00E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185645BDBM185645(US9161922, Table 1, Compound 11)
Affinity DataIC50: 1.10E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185639BDBM185639(US9161922, Table 1, Compound 5)
Affinity DataIC50: 1.30E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185648BDBM185648(US9161922, Table 2, Compound 3)
Affinity DataIC50: 1.35E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185640BDBM185640(US9161922, Table 1, Compound 6)
Affinity DataIC50: 2.00E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185643BDBM185643(US9161922, Table 1, Compound 9)
Affinity DataIC50: 2.40E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185657BDBM185657(US9161922, Table 3, Compound 2)
Affinity DataIC50: 9.00E+4nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185653BDBM185653(US9161922, Table 2, Compound 8)
Affinity DataIC50: 1.08E+5nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetHistamine oxidase(Arthrobacter globiformis)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185656BDBM185656(US9161922, Table 3, Compound 1)
Affinity DataIC50: 2.50E+5nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetAmine oxidase(Yeast)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185656BDBM185656(US9161922, Table 3, Compound 1)
Affinity DataIC50: 2.50E+5nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185637BDBM185637(US9161922, Table 1, Compound 2)
Affinity DataIC50: 5.00E+5nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 50026182BDBM50026182(3-Phenyl-prop-2-ynylamine | CHEMBL110611 | US91619...)
Affinity DataIC50: 7.00E+5nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185636BDBM185636(US9161922, Table 1, Compound 1)
Affinity DataIC50: 1.00E+6nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185656BDBM185656(US9161922, Table 3, Compound 1)
Affinity DataIC50: 1.80E+6nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185642BDBM185642(US9161922, Table 1, Compound 8)
Affinity DataIC50: 2.00E+6nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetAmine oxidase(Yeast)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185657BDBM185657(US9161922, Table 3, Compound 2)
Affinity DataIC50: 3.00E+6nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetHistamine oxidase(Arthrobacter globiformis)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185657BDBM185657(US9161922, Table 3, Compound 2)
Affinity DataIC50: 3.50E+6nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetAmine oxidase(Yeast)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185658BDBM185658(US9161922, Table 3, Compound 3)
Affinity DataIC50: 5.00E+6nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185654BDBM185654(US9161922, Table 2, Compound 9)
Affinity DataIC50: 6.50E+6nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent

TargetMembrane primary amine oxidase(Bovine)
Case Western Reserve University

US Patent
LigandChemical structure of BindingDB Monomer ID 185658BDBM185658(US9161922, Table 3, Compound 3)
Affinity DataIC50: 1.00E+7nMpH: 7.2 T: 2°CAssay Description:In the following Examples, 0.9 mL aliquots of a solution of candidate inhibitor in 100 mM potassium phosphate buffer, pH 7.2 was mixed bovine plasma ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details
US Patent