Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 7379
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 50069799BDBM50069799(CHEMBL3407579 | US9187441, 7M)
Affinity DataKi:  0.130nM ΔG°:  -55.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192221BDBM192221(US9187441, 7K)
Affinity DataKi:  0.150nM ΔG°:  -55.1kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192225BDBM192225(US9187441, 7P)
Affinity DataKi:  0.170nM ΔG°:  -54.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192217BDBM192217(US9187441, 7G)
Affinity DataKi:  0.200nM ΔG°:  -54.4kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192155BDBM192155(US9187441, 7E)
Affinity DataKi:  0.25nM ΔG°:  -53.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192161BDBM192161(US9187441, 7I)
Affinity DataKi:  0.300nM ΔG°:  -53.4kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192204BDBM192204(US9187441, 6M)
Affinity DataKi:  0.400nM ΔG°:  -52.7kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192213BDBM192213(US9187441, 7B)
Affinity DataKi:  0.450nM ΔG°:  -52.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192196BDBM192196(US9187441, 6E)
Affinity DataKi:  0.5nM ΔG°:  -52.2kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192228BDBM192228(US9187441, 7S)
Affinity DataKi:  0.700nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192151BDBM192151(US9187441, 7C)
Affinity DataKi:  0.810nM ΔG°:  -51.0kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192194BDBM192194(US9187441, 6C)
Affinity DataKi:  1.30nM ΔG°:  -49.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192241BDBM192241(US9187441, 6A)
Affinity DataKi:  1.5nM ΔG°:  -49.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192153BDBM192153(US9187441, 7D)
Affinity DataKi:  1.70nM ΔG°:  -49.2kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192229BDBM192229(US9187441, 7T)
Affinity DataKi:  1.80nM ΔG°:  -49.1kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192148BDBM192148(US9187441, 7A)
Affinity DataKi:  1.80nM ΔG°:  -49.1kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192202BDBM192202(US9187441, 6K)
Affinity DataKi:  2.10nM ΔG°:  -48.7kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192193BDBM192193(US9187441, 6B)
Affinity DataKi:  2.20nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192222BDBM192222(US9187441, 7L)
Affinity DataKi:  2.30nM ΔG°:  -48.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192216BDBM192216(US9187441, 7F)
Affinity DataKi:  2.30nM ΔG°:  -48.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192200BDBM192200(US9187441, 6I)
Affinity DataKi:  2.40nM ΔG°:  -48.4kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192207BDBM192207(US9187441, 6P)
Affinity DataKi:  2.5nM ΔG°:  -48.3kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192159BDBM192159(US9187441, 7H)
Affinity DataKi:  2.5nM ΔG°:  -48.3kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192198BDBM192198(US9187441, 6G)
Affinity DataKi:  3nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192195BDBM192195(US9187441, 6D)
Affinity DataKi:  3nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192227BDBM192227(US9187441, 7R)
Affinity DataKi:  3nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192226BDBM192226(US9187441, 7Q)
Affinity DataKi:  3nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192223BDBM192223(US9187441, 7N)
Affinity DataKi:  3.20nM ΔG°:  -47.7kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192224BDBM192224(US9187441, 7O)
Affinity DataKi:  3.20nM ΔG°:  -47.7kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192205BDBM192205(US9187441, 6N)
Affinity DataKi:  4.30nM ΔG°:  -47.0kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192201BDBM192201(US9187441, 6J)
Affinity DataKi:  4.5nM ΔG°:  -46.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192203BDBM192203(US9187441, 6L)
Affinity DataKi:  5nM ΔG°:  -46.6kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192220BDBM192220(US9187441, 7J)
Affinity DataKi:  5.70nM ΔG°:  -46.3kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192209BDBM192209(US9187441, 6R)
Affinity DataKi:  5.80nM ΔG°:  -46.2kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192211BDBM192211(US9187441, 6T)
Affinity DataKi:  5.80nM ΔG°:  -46.2kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192197BDBM192197(US9187441, 6F)
Affinity DataKi:  6nM ΔG°:  -46.1kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192208BDBM192208(US9187441, 6Q)
Affinity DataKi:  6.70nM ΔG°:  -45.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192206BDBM192206(US9187441, 6O)
Affinity DataKi:  6.80nM ΔG°:  -45.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192210BDBM192210(US9187441, 6S)
Affinity DataKi:  7nM ΔG°:  -45.8kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192199BDBM192199(US9187441, 6H)
Affinity DataKi:  10nM ΔG°:  -44.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 50014092BDBM50014092(CHEMBL3259830 | US9187441, 9l)
Affinity DataKi:  300nM ΔG°:  -36.6kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192240BDBM192240(US9187441, KK273)
Affinity DataKi:  400nM ΔG°:  -35.2kJ/molepH: 7.4 T: 2°CAssay Description:All NMR spectra were acquired at 298 K on a Bruker DRX 600 MHz spectrometer equipped with a cryoprobe. Typically, NMR samples contained 0.1-0.2 mM pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 50014092BDBM50014092(CHEMBL3259830 | US9187441, 9l)
Affinity DataKi:  400nM ΔG°:  -35.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192179BDBM192179(US9187441, 9n)
Affinity DataKi:  500nM ΔG°:  -35.4kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192178BDBM192178(US9187441, 9m)
Affinity DataKi:  600nM ΔG°:  -34.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 50014092BDBM50014092(CHEMBL3259830 | US9187441, 9l)
Affinity DataKi:  700nM ΔG°:  -34.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192244BDBM192244(US9187441, 11b)
Affinity DataKi:  700nM ΔG°:  -34.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192239BDBM192239(US9187441, KK271)
Affinity DataKi:  900nM ΔG°:  -33.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192182BDBM192182(US9187441, 9q)
Affinity DataKi:  900nM ΔG°:  -33.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Pittsburgh

US Patent
LigandChemical structure of BindingDB Monomer ID 192243BDBM192243(US9187441, 11a)
Affinity DataKi:  900nM ΔG°:  -33.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

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