Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 1744
LigandPNGBDBM337806((1E,3E)-1-(6-fluoropyridin-3-yl)-2-methylpent-1-en...)
Affinity DataIC50: 1.25E+3nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337809((1E,3E)-2-methyl-1-thien-3-ylpent-1-en-3-one oxime...)
Affinity DataIC50: 1.32E+3nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337811((1E,3E)-2-methyl-1-pyridin-4-ylpent-1-en-3-one oxi...)
Affinity DataIC50: 8.61E+3nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337807((1E,3E)-2-methyl-1-thien-2-ylpent-1-en-3-one oxime...)
Affinity DataIC50: 1.10E+4nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337810((1E,3E)-2-methyl-1-pyridin-3-ylpent-1-en-3-one oxi...)
Affinity DataIC50: 1.70E+4nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337808((1E,3E)-1-(6-methoxypyridin-3-yl)-2-methylpent-1-e...)
Affinity DataIC50: 2.34E+4nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337815((1E,3E)-2-methyl-1-[6-(trifluoromethyl)pyridin-3-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337816((1E,3E)-1-(isoquinolin-4-yl)-2-methylpent-1-en-3-o...)
Affinity DataIC50: 1.00E+5nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337813((1E,3E)-2-methyl-1-quinolin-3-ylpent-1-en-3-one ox...)
Affinity DataIC50: 1.00E+5nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337814((1E,3E)-2-methyl-1-(4-methylpyridin-3-yl)pent-1-en...)
Affinity DataIC50: 1.00E+5nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent

LigandPNGBDBM337812((1E,3E)-2-methyl-1-(6-methylpyridin-3-yl)pent-1-en...)
Affinity DataIC50: 1.00E+5nMAssay Description:Ca2+ influx was measured using a FLIPR calcium assay kit (R8033; Molecular Devices, Sunnyvale, Calif.). The Ca2+ indicator dye was dissolved in Hanks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2019
Entry Details
US Patent