Compile Data Set for Download or QSAR
Report error Found 132 Enz. Inhib. hit(s) with all data for entry = 1871
LigandChemical structure of BindingDB Monomer ID 50071821BDBM50071821(CHEMBL3410872 | US9783573, Example 6)
Affinity DataIC50: 3nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030280BDBM50030280(CHEMBL3339214 | US9783573, Example 10)
Affinity DataIC50: 3nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030270BDBM50030270(CHEMBL3339219 | US9783573, Example 23)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345205BDBM345205(US9783573, Example 55)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345172BDBM345172((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345175BDBM345175((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345152BDBM345152(US9783573, Example 2)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345168BDBM345168(US9783573, Example 18)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345213BDBM345213(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 5nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345176BDBM345176((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 5nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345207BDBM345207(US9783573, Example 57)
Affinity DataIC50: 6nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345215BDBM345215(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 6nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345171BDBM345171((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 6nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345209BDBM345209(N1-((35,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 7nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345205BDBM345205(US9783573, Example 55)
Affinity DataIC50: 9nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030270BDBM50030270(CHEMBL3339219 | US9783573, Example 23)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345207BDBM345207(US9783573, Example 57)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345214BDBM345214(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345209BDBM345209(N1-((35,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345163BDBM345163(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345170BDBM345170(US9783573, Example 20)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345206BDBM345206(US9783573, Example 56)
Affinity DataIC50: 12nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345161BDBM345161(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 12nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345163BDBM345163(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 12nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345172BDBM345172((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345215BDBM345215(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345214BDBM345214(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50071821BDBM50071821(CHEMBL3410872 | US9783573, Example 6)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030278BDBM50030278(CHEMBL3339215 | US9783573, Example 38)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345175BDBM345175((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345211BDBM345211(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345213BDBM345213(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345206BDBM345206(US9783573, Example 56)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345171BDBM345171((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345161BDBM345161(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 18nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345208BDBM345208(US9783573, Example 58)
Affinity DataIC50: 18nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345204BDBM345204(N4-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 21nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345199BDBM345199(US9783573, Example 49)
Affinity DataIC50: 22nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345210BDBM345210(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 22nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030280BDBM50030280(CHEMBL3339214 | US9783573, Example 10)
Affinity DataIC50: 23nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345168BDBM345168(US9783573, Example 18)
Affinity DataIC50: 23nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345201BDBM345201(N4-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 27nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345208BDBM345208(US9783573, Example 58)
Affinity DataIC50: 27nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345152BDBM345152(US9783573, Example 2)
Affinity DataIC50: 28nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345211BDBM345211(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 31nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345174BDBM345174((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 33nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345182BDBM345182(US9783573, Example 32)
Affinity DataIC50: 35nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345170BDBM345170(US9783573, Example 20)
Affinity DataIC50: 37nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345180BDBM345180(US9783573, Example 30)
Affinity DataIC50: 38nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 345202BDBM345202((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino)pro...)
Affinity DataIC50: 42nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
US Patent

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