Affinity DataKi: 0.690nMAssay Description:Ability of the compound to displace [125I]-HEAT from cloned human Alpha-1A adrenergic receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity of the compound against Alpha-1A adrenergic receptor in human prostatic tissueMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity of the compound against Alpha-1A adrenergic receptor in rat prostatic tissueMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 136nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 137nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 221nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 793nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.29E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.52E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.67E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.25E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.84E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair