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Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50008666
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075892(CHEMBL83753 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  330nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  380nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  580nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075906(4-[3-(3-Cyclopentyl-propyl)-2-oxo-imidazolidin-1-y...)
Affinity DataIC50:  760nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075911(4-[3-(3-Cyclopentyl-propyl)-2-oxo-2,3-dihydro-imid...)
Affinity DataIC50:  760nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075914(4-(3-Heptyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075902(4-[3-(2-Cyclohexyl-ethyl)-2-oxo-imidazolidin-1-yl]...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075910(4-[3-(3-Cyclohexyl-propyl)-2-oxo-imidazolidin-1-yl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075910(4-[3-(3-Cyclohexyl-propyl)-2-oxo-imidazolidin-1-yl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075913(4-{3-[3-(4-Chloro-phenyl)-propyl]-2-oxo-imidazolid...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075899(CHEMBL164401 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075908(CHEMBL166188 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075913(4-{3-[3-(4-Chloro-phenyl)-propyl]-2-oxo-imidazolid...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075896(4-(3-Hexyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-2...)
Affinity DataIC50:  2.30E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075906(4-[3-(3-Cyclopentyl-propyl)-2-oxo-imidazolidin-1-y...)
Affinity DataIC50:  2.40E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075914(4-(3-Heptyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075903(4-[3-(3,4-Difluoro-benzyl)-2-oxo-imidazolidin-1-yl...)
Affinity DataIC50:  3.50E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075902(4-[3-(2-Cyclohexyl-ethyl)-2-oxo-imidazolidin-1-yl]...)
Affinity DataIC50:  4.00E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075908(CHEMBL166188 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075904(CHEMBL165015 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075907(4-[3-(2-Cyclopentyl-ethyl)-2-oxo-imidazolidin-1-yl...)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075916(4-[3-(2,2-Dimethyl-hexyl)-2-oxo-imidazolidin-1-yl]...)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075903(4-[3-(3,4-Difluoro-benzyl)-2-oxo-imidazolidin-1-yl...)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075896(4-(3-Hexyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-2...)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075911(4-[3-(3-Cyclopentyl-propyl)-2-oxo-2,3-dihydro-imid...)
Affinity DataIC50:  5.30E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075898(4-(3-Butyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-2...)
Affinity DataIC50:  5.30E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075892(CHEMBL83753 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075915(CHEMBL79675 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  6.50E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075916(4-[3-(2,2-Dimethyl-hexyl)-2-oxo-imidazolidin-1-yl]...)
Affinity DataIC50:  8.50E+3nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075912(CHEMBL83754 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  9.00E+3nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075915(CHEMBL79675 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075905(CHEMBL349689 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075904(CHEMBL165015 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075899(CHEMBL164401 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075898(4-(3-Butyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-2...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075907(4-[3-(2-Cyclopentyl-ethyl)-2-oxo-imidazolidin-1-yl...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075912(CHEMBL83754 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075889(4-(3-Hexyl-2-oxo-2,3-dihydro-imidazol-1-yl)-N-{4-[...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075901(4-[3-(3,4-Difluoro-benzyl)-2-oxo-2,3-dihydro-imida...)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075889(4-(3-Hexyl-2-oxo-2,3-dihydro-imidazol-1-yl)-N-{4-[...)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075901(4-[3-(3,4-Difluoro-benzyl)-2-oxo-2,3-dihydro-imida...)
Affinity DataIC50:  2.70E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075900(CHEMBL434284 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  5.00E+4nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075900(CHEMBL434284 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  5.00E+4nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075905(CHEMBL349689 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataIC50:  1.00E+5nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075909(CHEMBL79915 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  1.00E+5nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075909(CHEMBL79915 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  1.00E+5nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075903(4-[3-(3,4-Difluoro-benzyl)-2-oxo-imidazolidin-1-yl...)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity towards Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075908(CHEMBL166188 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataEC50:  4.20nMAssay Description:Agonist activity towards Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075899(CHEMBL164401 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-...)
Affinity DataEC50:  85nMAssay Description:Agonist activity towards Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075901(4-[3-(3,4-Difluoro-benzyl)-2-oxo-2,3-dihydro-imida...)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity of the compound towards Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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