Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 5206
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50334460(RTI-229 | CHEMBL1643896 | ((1R,2S,3S,5S)-3-(4-iodo...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50006784(CHEMBL82946 | RTI-121 | 3-(4-Iodo-phenyl)-8-methyl...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85419(RTI-110)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50101075((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-methyl-8-a...)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50349799(CHEMBL1812745 | RTI-112)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85414(RTI-31)
Affinity DataKi:  1.12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22166(RTI 55, (exo,exo)-isomer, Iodine (125) labeled | R...)
Affinity DataKi:  1.26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50127390(RTI-147 | CHEMBL51355 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataKi:  1.38nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50006786(CHEMBL82093 | RTI-114 | 3-(4-Chloro-phenyl)-8-meth...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85416(RTI-51)
Affinity DataKi:  1.69nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50005539(RTI-32 | 8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85415(RTI-113)
Affinity DataKi:  1.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50101075((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-methyl-8-a...)
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85417(RTI-120)
Affinity DataKi:  3.26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85419(RTI-110)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22166(RTI 55, (exo,exo)-isomer, Iodine (125) labeled | R...)
Affinity DataKi:  4.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85419(RTI-110)
Affinity DataKi:  5.45nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50005572((3S,8R)-3-(4-Amino-phenyl)-8-methyl-8-aza-bicyclo[...)
Affinity DataKi:  9.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50349799(CHEMBL1812745 | RTI-112)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85416(RTI-51)
Affinity DataKi:  10.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50101075((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-methyl-8-a...)
Affinity DataKi:  17.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22166(RTI 55, (exo,exo)-isomer, Iodine (125) labeled | R...)
Affinity DataKi:  22.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22396(methyl (1R,2S,3S,5S)-8-methyl-3-phenyl-8-azabicycl...)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50349799(CHEMBL1812745 | RTI-112)
Affinity DataKi:  36.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85414(RTI-31)
Affinity DataKi:  37nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85416(RTI-51)
Affinity DataKi:  37.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85414(RTI-31)
Affinity DataKi:  44.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50005539(RTI-32 | 8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22166(RTI 55, (exo,exo)-isomer, Iodine (125) labeled | R...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22166(RTI 55, (exo,exo)-isomer, Iodine (125) labeled | R...)
Affinity DataKi:  66.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50006784(CHEMBL82946 | RTI-121 | 3-(4-Iodo-phenyl)-8-methyl...)
Affinity DataKi:  66.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22418(Cocaine (-) | methyl (1R,2R,3S,5S)-3-(benzoyloxy)-...)
Affinity DataKi:  102nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50005572((3S,8R)-3-(4-Amino-phenyl)-8-methyl-8-aza-bicyclo[...)
Affinity DataKi:  151nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50005539(RTI-32 | 8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50006784(CHEMBL82946 | RTI-121 | 3-(4-Iodo-phenyl)-8-methyl...)
Affinity DataKi:  285nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22166(RTI 55, (exo,exo)-isomer, Iodine (125) labeled | R...)
Affinity DataKi:  760nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50006786(CHEMBL82093 | RTI-114 | 3-(4-Chloro-phenyl)-8-meth...)
Affinity DataKi:  778nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22396(methyl (1R,2S,3S,5S)-8-methyl-3-phenyl-8-azabicycl...)
Affinity DataKi:  920nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50334460(RTI-229 | CHEMBL1643896 | ((1R,2S,3S,5S)-3-(4-iodo...)
Affinity DataKi:  990nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50006786(CHEMBL82093 | RTI-114 | 3-(4-Chloro-phenyl)-8-meth...)
Affinity DataKi:  1.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50334460(RTI-229 | CHEMBL1643896 | ((1R,2S,3S,5S)-3-(4-iodo...)
Affinity DataKi:  1.73E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22396(methyl (1R,2S,3S,5S)-8-methyl-3-phenyl-8-azabicycl...)
Affinity DataKi:  1.96E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85418(RIT-70)
Affinity DataKi:  2.07E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85415(RTI-113)
Affinity DataKi:  2.34E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85415(RTI-113)
Affinity DataKi:  2.93E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM22418(Cocaine (-) | methyl (1R,2R,3S,5S)-3-(benzoyloxy)-...)
Affinity DataKi:  3.83E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50127390(RTI-147 | CHEMBL51355 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataKi:  3.95E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50005572((3S,8R)-3-(4-Amino-phenyl)-8-methyl-8-aza-bicyclo[...)
Affinity DataKi:  5.11E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85417(RTI-120)
Affinity DataKi:  5.83E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM85418(RIT-70)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
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