Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50042027
TargetSolute carrier family 22 member 3(Human)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  1.40E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 2(Rat)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataKi:  2.80E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 2(Rat)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  3.90E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 1(Rat)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  1.40E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed