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Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50008900
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054245(5-Chloro-N-cyclopropylmethyl-2-methyl-N-propyl-N''...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054252(5-Bromo-N-cyclopropylmethyl-2-methyl-N-propyl-N'-(...)
Affinity DataKi:  2nMAssay Description:Ability to inhibit [125I]-CRH binding to human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054250(CHEMBL306482 | N-Cyclopropylmethyl-2,5-dimethyl-N-...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054248(2,5-Dimethyl-N,N-dipropyl-N'-(2,4,6-trichloro-phen...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054253(CHEMBL77716 | N-Cyclopropylmethyl-5-ethyl-2-methyl...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054225(CHEMBL306618 | N-Cyclopropylmethyl-6-methyl-N-prop...)
Affinity DataKi:  57nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054226(CHEMBL77391 | N,N-Diallyl-6-methyl-N'-(2,4,6-trime...)
Affinity DataKi:  115nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054230(6-Methyl-N,N-dipropyl-N'-(2,4,6-trimethyl-phenyl)-...)
Affinity DataKi:  130nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054246(CHEMBL77006 | N-Cyclopropylmethyl-2-methyl-N-propy...)
Affinity DataKi:  253nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054246(CHEMBL77006 | N-Cyclopropylmethyl-2-methyl-N-propy...)
Affinity DataKi:  253nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054216(CHEMBL307419 | N-Benzyl-6-methyl-N-propyl-N'-(2,4,...)
Affinity DataKi:  490nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054221(CHEMBL419636 | N,N-Dibutyl-6-methyl-N'-(2,4,6-trim...)
Affinity DataKi:  490nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054239(CHEMBL78035 | [4-(3,6-Dihydro-2H-pyridin-1-yl)-6-m...)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054219(CHEMBL305671 | N-Benzyl-N-butyl-6-methyl-N'-(2,4,6...)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054255(CHEMBL80806 | N-Cyclopropylmethyl-2-methyl-N-propy...)
Affinity DataKi:  1.39E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054223(CHEMBL307871 | N-Benzyl-N-ethyl-6-methyl-N'-(2,4,6...)
Affinity DataKi:  1.47E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054241(6-Methyl-N-(4-trifluoromethyl-benzyl)-N'-(2,4,6-tr...)
Affinity DataKi:  1.69E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054234(6,N-Dimethyl-N-phenethyl-N'-(2,4,6-trimethyl-pheny...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50078345(CHEMBL309789 | N-Cyclopropylmethyl-6-methyl-N-prop...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054235(CHEMBL78203 | N-Cyclopropylmethyl-6-ethyl-N-propyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed