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Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 5224
TargetSodium-dependent noradrenaline transporter(Human)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  4.21nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  5.74nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Bovine)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  6.01nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  7.36nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  8.54nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent noradrenaline transporter(Bovine)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  8.88nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNorepinephrine transporter(Rat)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  82.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Bovine)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  93.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  118nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Bovine)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM22418(Cocaine (-) | methyl (1R,2R,3S,5S)-3-(benzoyloxy)-...)
Affinity DataKi:  197nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  323nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNorepinephrine transporter(Rat)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  392nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Bovine)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  397nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNorepinephrine transporter(Rat)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM22418(Cocaine (-) | methyl (1R,2R,3S,5S)-3-(benzoyloxy)-...)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM81945(NSC_39484 | CHEMBL105891 | CHEMBL271379 | CHEMBL10...)
Affinity DataKi:  507nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Bovine)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM81945(NSC_39484 | CHEMBL105891 | CHEMBL271379 | CHEMBL10...)
Affinity DataKi:  570nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM81945(NSC_39484 | CHEMBL105891 | CHEMBL271379 | CHEMBL10...)
Affinity DataKi:  778nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM84342(EPINEPHRINE | 4-[1-hydroxy-2-(methylamino)ethyl]be...)
Affinity DataKi:  3.68E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Bovine)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM84342(EPINEPHRINE | 4-[1-hydroxy-2-(methylamino)ethyl]be...)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
The University of Queensland

Curated by PDSP Ki Database
LigandPNGBDBM84342(EPINEPHRINE | 4-[1-hydroxy-2-(methylamino)ethyl]be...)
Affinity DataKi:  6.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details
PubMed