Affinity DataKi: 21.3nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22.2nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 426nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 785nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.31E+3nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [125 I]AB-MECA from human Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.77E+3nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Displacement of [125 I]AB-MECA from human Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 4.77E+3nMAssay Description:Displacement of [3H]-CGS-21,680 from Adenosine A2A receptor of rat striatal membrane at 10e-4 microMMore data for this Ligand-Target Pair
Affinity DataKi: 5.93E+3nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.66E+3nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.64E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.35E+4nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 3.51E+4nMAssay Description:Displacement of [3H]-CGS-21,680 from Adenosine A2A receptor of rat striatal membrane at 10e-4 microMMore data for this Ligand-Target Pair
Affinity DataKi: 4.01E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.13E+4nMAssay Description:Displacement of [3H]-R-PIA from Adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 8.63E+4nMAssay Description:Displacement of [3H]-CGS-21,680 from Adenosine A2A receptor of rat striatal membrane at 10e-4 microMMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-CGS-21,680 from Adenosine A2A receptor of rat striatal membrane at 10e-4 microMMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-CGS-21,680 from Adenosine A2A receptor of rat striatal membrane at 10e-4 microMMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-R-PIA from Adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair