Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50009165
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080809(7-(4-Phenyl-3,6-dihydro-2H-pyridin-1-ylmethyl)-chr...)
Affinity DataKi:  4.40nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080797(7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataKi:  5.80nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080796(7-[4-(3-Chloro-4-methyl-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  6.90nMAssay Description:Binding affinity using [3H]spiperone displacement from cloned human Dopamine receptor D4.2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080794(7-[(2-p-Tolylamino-ethylamino)-methyl]-chromen-2-o...)
Affinity DataKi:  10nMAssay Description:Binding affinity using [3H]spiperone displacement from cloned human Dopamine receptor D4.2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080787(6-(4-p-Tolyl-piperazin-1-ylmethyl)-chromen-2-one |...)
Affinity DataKi:  11nMAssay Description:Binding affinity using [3H]spiperone displacement from cloned human Dopamine receptor D4.2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080810(7-[4-(3,4-Dimethyl-phenyl)-piperazin-1-ylmethyl]-c...)
Affinity DataKi:  14nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080798(7-{[2-(4-Chloro-phenylamino)-ethylamino]-methyl}-c...)
Affinity DataKi:  14nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080788(7-(4-o-Tolyl-piperazin-1-ylmethyl)-chromen-2-one |...)
Affinity DataKi:  16nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080800(7-{[2-(3-Chloro-4-methyl-phenylamino)-ethylamino]-...)
Affinity DataKi:  16nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080790(7-(4-p-Tolyl-piperazin-1-ylmethyl)-chromen-2-one |...)
Affinity DataKi:  17nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080786(7-(4-Phenyl-piperidin-1-ylmethyl)-chromen-2-one | ...)
Affinity DataKi:  19nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080806(7-{[2-(3,4-Dimethyl-phenylamino)-ethylamino]-methy...)
Affinity DataKi:  21nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080808(7-(4-Phenyl-piperazin-1-ylmethyl)-chromen-2-one | ...)
Affinity DataKi:  27nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080801(6-(4-Phenyl-piperazin-1-ylmethyl)-chromen-2-one | ...)
Affinity DataKi:  30nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080805(7-[(3-Phenylamino-propylamino)-methyl]-chromen-2-o...)
Affinity DataKi:  31nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080795(7-(4-m-Tolyl-piperazin-1-ylmethyl)-chromen-2-one |...)
Affinity DataKi:  32nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080792(7-[(2-Phenoxy-ethylamino)-methyl]-chromen-2-one | ...)
Affinity DataKi:  43nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080812(7-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-chrom...)
Affinity DataKi:  59nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080793(6-(4-o-Tolyl-piperazin-1-ylmethyl)-chromen-2-one |...)
Affinity DataKi:  63nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080799(6-(4-m-Tolyl-piperazin-1-ylmethyl)-chromen-2-one |...)
Affinity DataKi:  74nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080804(7-[4-(4-Methoxy-phenyl)-piperazin-1-ylmethyl]-chro...)
Affinity DataKi:  75nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080791(7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-chrom...)
Affinity DataKi:  93nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080802(7-[4-(4-tert-Butyl-phenyl)-piperazin-1-ylmethyl]-c...)
Affinity DataKi:  227nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080803(6-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataKi:  311nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080811(7-{[Ethyl-(2-phenylamino-ethyl)-amino]-methyl}-chr...)
Affinity DataKi:  410nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080797(7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataKi:  424nMAssay Description:Compound was tested for binding affinity using [3H]spiperone against cloned human Dopamine receptor D3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080789(7-{[2-(Ethyl-phenyl-amino)-ethylamino]-methyl}-chr...)
Affinity DataKi:  2.66E+3nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080797(7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataKi:  2.67E+3nMAssay Description:Compound was tested for binding affinity using [3H]prazosin against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080807(7-(4-Benzyl-piperazin-1-ylmethyl)-chromen-2-one | ...)
Affinity DataKi:  2.70E+3nMAssay Description:Compound was tested for the inhibition of [3H]thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080797(7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataKi:  3.71E+3nMAssay Description:Compound was tested for binding affinity using [3H]8-OH-DPAT against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(BOVINE)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080797(7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataKi: >4.35E+3nMAssay Description:Compound was tested for binding affinity using [3H]ketanserin against 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080797(7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataKi: >4.70E+3nMAssay Description:Compound was tested for binding affinity using [3H]MK-912 against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080797(7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-on...)
Affinity DataIC50:  1.30nMAssay Description:Compound was tested for the inhibition of [3H]-thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080796(7-[4-(3-Chloro-4-methyl-phenyl)-piperazin-1-ylmeth...)
Affinity DataIC50:  5.40nMAssay Description:Compound was tested for the inhibition of [3H]-thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080794(7-[(2-p-Tolylamino-ethylamino)-methyl]-chromen-2-o...)
Affinity DataIC50:  98nMAssay Description:Compound was tested for the inhibition of [3H]-thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080787(6-(4-p-Tolyl-piperazin-1-ylmethyl)-chromen-2-one |...)
Affinity DataIC50: >1.00E+3nMAssay Description:Compound was tested for the inhibition of [3H]-thymidine uptake in CHO p-5 cells transfected with human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed