Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50009429
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083552BDBM50083552(1,9-di{4-[5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  0.0190nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083561BDBM50083561(1-{4-[5-amino(imino)methylbenzo[b]thiophen-2-ylcar...)
Affinity DataKi:  0.0280nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083556BDBM50083556(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  0.0290nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083541BDBM50083541(1-{4-[5-amino(imino)methyl-4,5,6,7-tetrahydrothien...)
Affinity DataKi:  0.0460nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083548BDBM50083548(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  0.0570nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217306BDBM50217306(CHEMBL112049)
Affinity DataKi:  0.120nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083549BDBM50083549(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217313BDBM50217313(CHEMBL110856)
Affinity DataKi:  60nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217310BDBM50217310(CHEMBL109688)
Affinity DataKi:  67nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217308BDBM50217308(CHEMBL424436)
Affinity DataKi:  210nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217305BDBM50217305(CHEMBL323935)
Affinity DataKi:  460nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217315BDBM50217315(CHEMBL30862)
Affinity DataKi:  970nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217312BDBM50217312(CHEMBL324918)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083563BDBM50083563(1-{4-[5-amino(imino)methylaminobenzo[b]furan-2-ylc...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217317BDBM50217317(CHEMBL109903)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083562BDBM50083562(2-(4-{2-[4-(5-Carbamimidoyl-benzofuran-2-carbonyl)...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217309BDBM50217309(CHEMBL111451)
Affinity DataKi:  6.60E+3nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217314BDBM50217314(CHEMBL112894)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217307BDBM50217307(CHEMBL112900)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083556BDBM50083556(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083561BDBM50083561(1-{4-[5-amino(imino)methylbenzo[b]thiophen-2-ylcar...)
Affinity DataKi:  2.20E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217316BDBM50217316(CHEMBL113084)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083547BDBM50083547(1,5-di(4-(5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083563BDBM50083563(1-{4-[5-amino(imino)methylaminobenzo[b]furan-2-ylc...)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083557BDBM50083557(N-Benzyl-2-(4-{2-[4-(5-carbamimidoyl-benzofuran-2-...)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083541BDBM50083541(1-{4-[5-amino(imino)methyl-4,5,6,7-tetrahydrothien...)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083548BDBM50083548(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083542BDBM50083542(1,5-di{4-[5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083543BDBM50083543(1,4-di{4-[5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  5.10E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50217311BDBM50217311(CHEMBL109660)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083553BDBM50083553(1,3-di{4-[5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  8.20E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083545BDBM50083545(1,7-di{4-[5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  8.50E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083549BDBM50083549(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  8.80E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083552BDBM50083552(1,9-di{4-[5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  2.30E+5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed