Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50009454
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083743BDBM50083743(1N-[1-amino(imino)methyl-6-hydroxy-(5S)-tetrahydro...)
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083747BDBM50083747(Cinnoline-4-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 4.20nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083756BDBM50083756(Isoquinoline-1-carboxylic acid ((R)-3-{[((S)-1-car...)
Affinity DataIC50: 4.90nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083754BDBM50083754(Pyrazine-2-carboxylic acid ((R)-3-{[((S)-1-carbami...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083747BDBM50083747(Cinnoline-4-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 5.60nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083744BDBM50083744(N-((R)-3-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 6.10nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083745BDBM50083745(5-Bromo-N-((R)-3-{[((S)-1-carbamimidoyl-2-hydroxy-...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083750BDBM50083750(Quinoline-3-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083751BDBM50083751(Pyrazine-2-carboxylic acid ((R)-4-{[((S)-1-carbami...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083742BDBM50083742({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083749BDBM50083749(Pyridine-2-carboxylic acid ((R)-3-{[((S)-1-carbami...)
Affinity DataIC50: 21nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083744BDBM50083744(N-((R)-3-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 27nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083753BDBM50083753({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083740BDBM50083740(((R)-3-[(5-Bromo-pyridine-3-carbonyl)-amino]-1-{[(...)
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083739BDBM50083739({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083746BDBM50083746(Quinoline-2-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 44nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083746BDBM50083746(Quinoline-2-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 59nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083741BDBM50083741({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 75nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083743BDBM50083743(1N-[1-amino(imino)methyl-6-hydroxy-(5S)-tetrahydro...)
Affinity DataIC50: 75nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083752BDBM50083752(N-((R)-3-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 79nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083756BDBM50083756(Isoquinoline-1-carboxylic acid ((R)-3-{[((S)-1-car...)
Affinity DataIC50: 98nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083739BDBM50083739({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 106nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083753BDBM50083753({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 106nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083750BDBM50083750(Quinoline-3-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 111nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083748BDBM50083748(Pyrazine-2-carboxylic acid ((R)-2-{[((S)-1-carbami...)
Affinity DataIC50: 152nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083745BDBM50083745(5-Bromo-N-((R)-3-{[((S)-1-carbamimidoyl-2-hydroxy-...)
Affinity DataIC50: 160nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083754BDBM50083754(Pyrazine-2-carboxylic acid ((R)-3-{[((S)-1-carbami...)
Affinity DataIC50: 166nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083742BDBM50083742({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 169nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083749BDBM50083749(Pyridine-2-carboxylic acid ((R)-3-{[((S)-1-carbami...)
Affinity DataIC50: 223nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083750BDBM50083750(Quinoline-3-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 250nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083748BDBM50083748(Pyrazine-2-carboxylic acid ((R)-2-{[((S)-1-carbami...)
Affinity DataIC50: 311nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083738BDBM50083738({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 313nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083740BDBM50083740(((R)-3-[(5-Bromo-pyridine-3-carbonyl)-amino]-1-{[(...)
Affinity DataIC50: 313nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083751BDBM50083751(Pyrazine-2-carboxylic acid ((R)-4-{[((S)-1-carbami...)
Affinity DataIC50: 324nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083741BDBM50083741({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 346nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083744BDBM50083744(N-((R)-3-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 367nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083754BDBM50083754(Pyrazine-2-carboxylic acid ((R)-3-{[((S)-1-carbami...)
Affinity DataIC50: 521nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083750BDBM50083750(Quinoline-3-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 537nMAssay Description:In vitro inhibition of human Thrombin (FIIa).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083752BDBM50083752(N-((R)-3-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 561nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083751BDBM50083751(Pyrazine-2-carboxylic acid ((R)-4-{[((S)-1-carbami...)
Affinity DataIC50: 673nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083747BDBM50083747(Cinnoline-4-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083756BDBM50083756(Isoquinoline-1-carboxylic acid ((R)-3-{[((S)-1-car...)
Affinity DataIC50: 730nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083745BDBM50083745(5-Bromo-N-((R)-3-{[((S)-1-carbamimidoyl-2-hydroxy-...)
Affinity DataIC50: 1.06E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083742BDBM50083742({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 1.14E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083749BDBM50083749(Pyridine-2-carboxylic acid ((R)-3-{[((S)-1-carbami...)
Affinity DataIC50: 1.14E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083746BDBM50083746(Quinoline-2-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 1.27E+3nMAssay Description:In vitro inhibition of human Thrombin (FIIa).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083746BDBM50083746(Quinoline-2-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 1.44E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083748BDBM50083748(Pyrazine-2-carboxylic acid ((R)-2-{[((S)-1-carbami...)
Affinity DataIC50: 1.48E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083747BDBM50083747(Cinnoline-4-carboxylic acid ((R)-3-{[((S)-1-carbam...)
Affinity DataIC50: 1.77E+3nMAssay Description:In vitro inhibition of human Thrombin (FIIa).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083753BDBM50083753({(R)-1-{[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-...)
Affinity DataIC50: 2.03E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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